Patent · US Active

Covalent inhibitors of K-Ras G12C

US9926267B2 · kind B2 · utility

37Cited by
18References
35Claims
0Family size

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Key dates

Filing dateNov 5, 2015
Grant dateMar 27, 2018
Priority date
Expiry dateNov 5, 2035

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG01N33/58
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Irreversible inhibitors of G12C mutant K-Ras protein are provided. Also disclosed are methods to modulate the activity of G12C mutant K-Ras protein and methods of treatment of disorders mediated by G12C mutant K-Ras protein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.