Patent · US Active

Pharmaceutical compounds

US9943519B2 · kind B2 · utility

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18References
5Claims
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Key dates

Filing dateJun 26, 2014
Grant dateApr 17, 2018
Priority date
Expiry dateJun 26, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of Formulae Ia, and stereoisomers, geometric isomers, tautomers, solvates, metabolites and pharmaceutically acceptable salts thereof, are useful for inhibiting lipid kinases including PI3K, and for treating disorders such as cancer mediated by lipid kinases. Methods of using compounds of Formula Ia for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.