Antony Bigot
23Patents
5h-index
50Co-inventors
68Inventor score
Filing activity: Apr 19, 2001 → Nov 3, 2016
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US7265111B2 | Adenosine analogues and their use as pharmaceutical agents | Chemistry; Metallurgy | 81 | Expired |
| US6531497B1 | Epothilone derivatives and their synthesis and use | Emerging Cross-Sectional Technologies | 26 | Expired |
| US6841562B2 | Quinolylpropylpiperidine derivatives, intermediates and compositions containing them, and preparation therefor | Emerging Cross-Sectional Technologies | 15 | Expired |
| US7232834B2 | Quinolylpropylpiperidine derivatives, intermediates and compositions containing them, and preparation therefor | Emerging Cross-Sectional Technologies | 9 | Expired |
| US7232833B2 | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them | Chemistry; Metallurgy | 6 | Expired |
| US6451821B1 | Use of 2-aminothiazoline derivatives as inhibitors of inducible no-synthase | Chemistry; Metallurgy | 3 | Expired |
| US7589117B2 | Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them | Human Necessities | 2 | Active |
| US6699867B2 | Use of 2-amino-thiazoline derivatives as inhibitors of inducible NO-synthase | Chemistry; Metallurgy | 2 | Expired |
| US7078428B2 | Isoindolone derivatives, preparation process and intermediates of this process, their use as medicaments, and pharmaceutical compositions comprising them | Human Necessities | 2 | Expired |
| US8314244B2 | Method for preparing activated esters | Chemistry; Metallurgy | 1 | Active |
| US10941139B2 | Cryptophycin compounds and conjugates, their preparation and their therapeutic use | Chemistry; Metallurgy | 1 | Active |
| US6420566B2 | Pharmaceutical compositions containing a 4, 5-dihydro-1, 3-thiazol-2-ylamine derivative, novel derivatives and preparation thereof | Chemistry; Metallurgy | 1 | Expired |
| US7348434B2 | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them | Chemistry; Metallurgy | 1 | Expired |
| US7579366B2 | Epothilone derivatives and their synthesis and use | Emerging Cross-Sectional Technologies | 1 | Expired |
| US8865906B2 | Process for the preparation of a compound useful as an inhibitor of TAFIa | Chemistry; Metallurgy | 0 | Active |
| US6699895B2 | 2-aminothiazoline derivatives and process for preparing the same | Chemistry; Metallurgy | 0 | Expired |
| US7227022B2 | Use of 2-amino-thiazoline derivatives as inhibitors of inducible no-synthase | Chemistry; Metallurgy | 0 | Expired |
| US6953796B2 | Use of 2-amino-thiazoline derivatives as inhibitors of inducible No-synthase | Chemistry; Metallurgy | 0 | Expired |
| US8119813B2 | Method for preparing enantiomerically enriched N-carboxyanhydride | Chemistry; Metallurgy | 0 | Active |
| US6872740B2 | Use of 2-amino-4-heteroarylethyl-thiazoline derivatives as inhibitors of inducible no-synthase | Chemistry; Metallurgy | 0 | Expired |
| US7884123B2 | Substituted thieno[2,3-c]pyrazoles, process for preparing them, compositions containing them, and use thereof | Human Necessities | 0 | Active |
| US8207355B2 | Method for preparing azetidine derivatives | Chemistry; Metallurgy | 0 | Active |
| US6762196B2 | Use of 2-amino-4-pyridylmethyl-thiazoline derivatives as inhibitors of inducible no-synthase | Chemistry; Metallurgy | 0 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.