Patent · US Expired

Cycloalkyl tachykinin receptor antagonists

US5750549A · kind A · utility

44Cited by
8References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 15, 1996
Grant dateMay 12, 1998
Priority date
Expiry dateOct 15, 2016

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention is directed to certain novel compounds represented by structural formula I: ##STR1## or a pharmaceutically acceptable salt thereof, wherein R.sup.3, R.sup.6, R.sup.7, R.sup.8, R.sup.11, R.sup.12, R.sup.13, A, Q, W, X, Y, Z and n are defined herein. The invention is also concerned with pharmaceutical formulations comprising these novel compounds as active ingredients and the use of the novel compounds and their formulations in the treatment of certain disorders. The compounds of this invention are tachykinin receptor antagonists and are useful in the treatment of inflammatory diseases, pain or migraine, asthma and emesis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.