Inventor · Hitchin, GB

Michael Alistair O'Brien

25Patents
11h-index
43Co-inventors
71Inventor score

Filing activity: Jul 5, 2004 → Jun 17, 2020

Most-cited inventions

PatentTitleAreaCited byStatus
US9670183B2 Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 30 Active
US7977477B2 Benzimidazole derivatives and their use as protein kinase inhibitors Chemistry; Metallurgy 26 Active
US8895745B2 Bicyclic heterocyclic compounds as FGFR inhibitors Chemistry; Metallurgy 24 Active
US9593106B2 Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists Chemistry; Metallurgy 20 Active
US10196380B2 Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 16 Active
US9926297B2 Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor agonists Chemistry; Metallurgy 15 Active
US7385059B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 15 Expired
US8106057B2 Dihydroxyphenyl isoindolylmethanones Chemistry; Metallurgy 12 Active
US10385039B2 Bicyclic aza compounds as muscarnic M1 receptor and/or M4 receptor antagonists Chemistry; Metallurgy 12 Active
US8101648B2 Hydroxybenzamide derivatives and their use as inhibitors of HSP90 Chemistry; Metallurgy 12 Active
US7754725B2 Dihydroxyphenyl isoindolymethanones Chemistry; Metallurgy 12 Active
US10689368B2 Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor Chemistry; Metallurgy 11 Active
US10961225B2 Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor Chemistry; Metallurgy 10 Active
US10030012B2 Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists Chemistry; Metallurgy 9 Active
US8513276B2 Imidazo[1,2-a]pyridine compounds for use in treating cancer Chemistry; Metallurgy 6 Active
US8530469B2 Therapeutic combinations of hydroxybenzamide derivatives as inhibitors of HSP90 Chemistry; Metallurgy 6 Active
US7745638B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 6 Active
US8080666B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 5 Active
US7825140B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 4 Active
US8779132B2 Pharmaceutical compounds Chemistry; Metallurgy 2 Active
US8779147B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 2 Active
US12227521B2 CGRP antagonist compounds Chemistry; Metallurgy 0 Active
US12344621B2 CGRP antagonist compounds Chemistry; Metallurgy 0 Active
US9051278B2 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators Chemistry; Metallurgy 0 Active
US9914719B2 Hydroxybenzamide derivatives and their use as inhibitors of HSP90 Chemistry; Metallurgy 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.