Stacey Shepard
58Patents
23h-index
37Co-inventors
84Inventor score
Filing activity: Dec 12, 2006 → Feb 1, 2024
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US7598257B2 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 224 | Active |
| US8158616B2 | Azetidine and cyclobutane derivatives as JAK inhibitors | Emerging Cross-Sectional Technologies | 133 | Active |
| US7834022B2 | Metabolites of the Janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Chemistry; Metallurgy | 120 | Active |
| US8486902B2 | Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d] pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Chemistry; Metallurgy | 106 | Active |
| US8716303B2 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 101 | Active |
| US8415362B2 | Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 100 | Active |
| US8933085B2 | Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors | Chemistry; Metallurgy | 90 | Active |
| US8420629B2 | Azetidine and cyclobutane derivatives as JAK inhibitors | Emerging Cross-Sectional Technologies | 90 | Active |
| US8530485B2 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 84 | Active |
| US8541425B2 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 80 | Active |
| US8748401B2 | Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Chemistry; Metallurgy | 75 | Active |
| US8889697B2 | Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Chemistry; Metallurgy | 75 | Active |
| US8933086B2 | Heteroaryl substituted pyrrolo[2,3-B]pyridines and pyrrolo[2,3-B]pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 66 | Active |
| US8946245B2 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 65 | Active |
| US9079912B2 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase inhibitors | Chemistry; Metallurgy | 65 | Active |
| US9334274B2 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 52 | Active |
| US9206187B2 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase | Chemistry; Metallurgy | 50 | Active |
| US9249145B2 | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | Human Necessities | 42 | Active |
| US9974790B2 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 36 | Active |
| US10138248B2 | Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-γ inhibitors | Chemistry; Metallurgy | 32 | Active |
| US9309246B2 | Tricyclic heterocycles as BET protein inhibitors | Human Necessities | 31 | Active |
| US9193733B2 | Piperidinylcyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors | Chemistry; Metallurgy | 30 | Active |
| US10398699B2 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 27 | Active |
| US9662335B2 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors | Chemistry; Metallurgy | 23 | Active |
| US9777003B2 | Tricyclic heterocycles as bet protein inhibitors | Human Necessities | 23 | Active |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.