Patent · US Expired

Process for preparing morpholine tachykinin receptor antagonists

US5637699A · kind A · utility

27Cited by
14References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 22, 1995
Grant dateJun 10, 1997
Priority date
Expiry dateMay 22, 2015

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Substituted heterocycles of the general structural formula: ##STR1## are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, asthma and emesis, and calcium channel blockers useful in the treatment of cardiovascular conditions such as angina, hypertension or ischemia.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.