Jeffrey J. Hale
42Patents
14h-index
74Co-inventors
80Inventor score
Filing activity: Sep 30, 1992 → May 6, 2011
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US5719147A | Morpholine and thiomorpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 83 | Expired |
| US5691336A | Morpholine compounds are prodrugs useful as tachykinin receptor antagonists | Chemistry; Metallurgy | 79 | Expired |
| US6166037A | Pyrrolidine and piperidine modulators of chemokine receptor activity | Chemistry; Metallurgy | 57 | Expired |
| US5750549A | Cycloalkyl tachykinin receptor antagonists | Chemistry; Metallurgy | 44 | Expired |
| US5877191A | Phenyl spiroethercycloalkyl tachykinin receptor antagonists | Chemistry; Metallurgy | 35 | Expired |
| US5512570A | Treatment of emesis with morpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 31 | Expired |
| US5780467A | Morpholine compounds are prodrugs useful as tachykinin receptor antagonists | Chemistry; Metallurgy | 30 | Expired |
| US5637699A | Process for preparing morpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 27 | Expired |
| US5716942A | Treatment of migraine with morpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 26 | Expired |
| US6248755A | Pyrrolidine modulators of chemokine receptor activity | Chemistry; Metallurgy | 24 | Expired |
| US5869496A | Spiro-substituted azacycles as tachykinin receptor antagonists | Chemistry; Metallurgy | 21 | Expired |
| US7605171B2 | (3,4-disubstituted)propanoic carboxylates as S1P (Edg) receptor agonists | Chemistry; Metallurgy | 20 | Expired |
| US7309721B2 | Aminoalkylphosphonates and related compounds as Edg receptor agonists | Chemistry; Metallurgy | 18 | Expired |
| US7351725B2 | N-(benzyl)aminoalkylcarboxylates, phosphinates, phosphonates and tetrazoles as Edg receptor agonists | Chemistry; Metallurgy | 17 | Expired |
| US7220734B2 | 1-(amino)indanes and (1,2-dihydro-3-amino)-benzofurans, benzothiophenes and indoles as Edg receptor agonists | Chemistry; Metallurgy | 14 | Expired |
| US5591737A | Substituted azetidinones as anti-inflammatory and antidegenerative agents | Chemistry; Metallurgy | 13 | Expired |
| US7479504B2 | Edg receptor agonists | Chemistry; Metallurgy | 13 | Expired |
| US7199142B2 | 1-((5-aryl-1,2,4-oxadiazol-3-yl) benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl) pyrrolidine-3-carboxylates as edg receptor agonists | Chemistry; Metallurgy | 12 | Expired |
| US6399619B1 | Pyrrolidine modulators of chemokine receptor activity | Chemistry; Metallurgy | 12 | Expired |
| US8354403B2 | Pyrrolidine derived beta 3 adrenergic receptor agonists | Chemistry; Metallurgy | 12 | Active |
| US5872116A | Morpholine and thiomorpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 11 | Expired |
| US5747485A | Substituted azetidiones as anti-inflammatory and antidegenerative agents | Human Necessities | 10 | Expired |
| US6048859A | Morpholine and thiomorpholine tachykinin receptor antagonists | Chemistry; Metallurgy | 9 | Expired |
| US7999107B2 | Substituted pyrano[2,3-B]pyridine derivatives as cannabinoid-1 receptor modulators | Chemistry; Metallurgy | 8 | Active |
| US6265434A | Pyrrolidine modulators of chemokine receptor activity | Chemistry; Metallurgy | 7 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.