Spiro-substituted azacycles as tachykinin receptor antagonists
US5869496A · kind A · utility
21Cited by
3References
16Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Jul 11, 1995 |
| Grant date | Feb 9, 1999 |
| Priority date | — |
| Expiry date | Jul 11, 2015 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D491/10
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Disclosed are spiro-substituted azacycles of formula (I), are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, emesis and asthma. In particular compounds of formula (I) are shown to be neurokinin antagonists. ##STR1##
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.