Patent · US Expired

Isoxazole compositions useful as inhibitors of ERK

US6495582B1 · kind B1 · utility

55Cited by
2References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 14, 2001
Grant dateDec 17, 2002
Priority date
Expiry dateSep 14, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are compounds that are useful as protein kinase inhibitors, especially inhibitors of ERK, having the formula: where A, B, R1, R2, T and Ht are described in the specification. The compounds are useful for treating diseases in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.