Inventor · Bedford, MA, US

Michael Hale

48Patents
18h-index
56Co-inventors
84Inventor score

Filing activity: Dec 24, 1997 → Nov 22, 2022

Most-cited inventions

PatentTitleAreaCited byStatus
US6784195B2 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 126 Expired
US6528509B1 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 100 Expired
US6743791B2 Heterocyclic inhibitors of ERK2 and uses thereof Chemistry; Metallurgy 78 Expired
US7253187B2 Heterocyclic inhibitors of ERK2 and uses thereof Chemistry; Metallurgy 69 Expired
US6495582B1 Isoxazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 55 Expired
US7304061B2 Heterocyclic inhibitors of ERK2 and uses thereof Chemistry; Metallurgy 55 Expired
US7345054B2 Heterocyclic inhibitors of ERK2 and uses thereof Chemistry; Metallurgy 52 Expired
US6593357B1 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 49 Expired
US6699865B2 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 44 Expired
US6949580B2 Pyrazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 40 Expired
US7056944B2 Pyrazole compositions useful as inhibitors of erk Chemistry; Metallurgy 38 Expired
US6319946A Inhibitors of aspartyl protease Chemistry; Metallurgy 35 Expired
US7304071B2 Protein kinase inhibitors and uses thereof Chemistry; Metallurgy 33 Expired
US7244735B2 Heterocyclic protein kinase inhibitors and uses thereof Chemistry; Metallurgy 29 Expired
US7407962B2 Heteroaryl compounds useful as inhibitors or protein kinases Chemistry; Metallurgy 26 Expired
US7501415B2 Selective inhibitors of ERK protein kinase and uses thereof Human Necessities 24 Active
US7456190B2 Compositions useful as protein kinase inhibitors Chemistry; Metallurgy 23 Expired
US7358258B2 Prodrugs of an ERK protein kinase inhibitor Human Necessities 23 Expired
US7354939B2 Pyrrole inhibitors of ERK protein kinase, synthesis thereof and intermediates thereto Chemistry; Metallurgy 17 Expired
US6436989B1 Prodrugs of aspartyl protease inhibitors Chemistry; Metallurgy 17 Expired
US6649640B2 Isoxazole compositions useful as inhibitors of ERK Chemistry; Metallurgy 15 Expired
US7169798B2 Inhibitors of c-Jun N terminal kinases (JNK) and other protein kinases Chemistry; Metallurgy 14 Expired
US6875789B2 Pyrazole-derived kinase inhibitors and uses thereof Chemistry; Metallurgy 11 Expired
US6750239B2 Pyrazole-derived kinase inhibitors and uses thereof Human Necessities 9 Expired
US6693108B2 Inhibitors of c-JUN N terminal kinases (JNK) and other protein kinases Chemistry; Metallurgy 8 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.