Patent · US Expired

Pyrazole compositions useful as inhibitors of ERK

US6784195B2 · kind B2 · utility

126Cited by
3References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 5, 2001
Grant dateAug 31, 2004
Priority date
Expiry dateMar 28, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are compounds that are useful as protein kinase inhibitors having the formula: where R1, R2, T and Ht are described in the specification. The compounds are useful for treating disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.