Patent assignee · BE · COMPANY

Janssen Pharmaceutica NA

1,055Patents
341Active
1,055Granted
52Portfolio score

Filing activity: Jun 21, 1974 → Sep 8, 2021 · 268 expiring within 5 years

Most-cited patents

PatentTitleAreaCited byStatus
US4837168A Immunoassay using colorable latex particles Emerging Cross-Sectional Technologies 205 Expired
US6407079B1 Pharmaceutical compositions containing drugs which are instable or sparingly soluble in water and methods for their preparation Human Necessities 166 Expired
US4804663A 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles Chemistry; Metallurgy 116 Expired
US6667060B1 Pregelatinized starch in a controlled release formulation Human Necessities 113 Expired
US7514445B2 Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors) Chemistry; Metallurgy 112 Expired
US4764604A Derivatives of gamma-cyclodextrin Performing Operations; Transporting 110 Expired
US7541367B2 3-benzoimidazolyl-pyrazolopyridines useful in treating kinase disorders Human Necessities 98 Active
US4775636A Blot overlay assay using colloidal metal particles Emerging Cross-Sectional Technologies 94 Expired
US5041448A (4-piperidinylmethyl and -hetero) purines Chemistry; Metallurgy 89 Expired
US4335127A Piperidinylalkyl quinazoline compounds, composition and method of use Chemistry; Metallurgy 85 Expired
US5258380A (4-piperidinylmethyl and -hetero)purines Chemistry; Metallurgy 84 Expired
US4962115A Novel N-(3-hydroxy-4-piperidinyl)benzamide derivatives Chemistry; Metallurgy 78 Expired
US7125879B2 HIV inhibiting pyrimidines derivatives Chemistry; Metallurgy 76 Expired
US4079062A Triazole derivatives Chemistry; Metallurgy 73 Expired
US6987110B2 Substituted pyrrolines as kinase inhibitors Chemistry; Metallurgy 71 Expired
US5246915A Method for controlling weeds Human Necessities 66 Expired
US5057525A Novel N-(3-hydroxy-4-piperidinyl) benzamide derivatives Chemistry; Metallurgy 60 Expired
US5158952A 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use Chemistry; Metallurgy 60 Expired
US4695575A 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines Chemistry; Metallurgy 57 Expired
US6544559B2 Microencapsulated 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles Human Necessities 57 Expired
US4267179A Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidaz oles and 1H-1,2,4-triazoles Chemistry; Metallurgy 56 Expired
US6037350A Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quionlinone derivatives Emerging Cross-Sectional Technologies 55 Expired
US6169096A Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives Emerging Cross-Sectional Technologies 54 Expired
US6207142A Compositions containing an antifungal and a cationic agent Human Necessities 54 Expired
US4144346A Novel 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles Chemistry; Metallurgy 54 Expired

Source: USPTO / EPO open patent data. Counts and citation impact are objective bibliographic measures.