Inventor · West Chester, PA, US

Gregory R. Ott

27Patents
6h-index
73Co-inventors
72Inventor score

Filing activity: Mar 16, 2001 → Apr 29, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US6740649B2 Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- &agr; converting enzyme (TACE) Chemistry; Metallurgy 15 Expired
US8148391B2 Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-Met inhibitors Chemistry; Metallurgy 11 Active
US9604994B2 Thienopyrimidine inhibitors of atypical protein kinase C Chemistry; Metallurgy 11 Active
US6984648B2 Cyclic β-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-α Chemistry; Metallurgy 10 Expired
US6743807B2 Cyclic &bgr;-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-&agr; Chemistry; Metallurgy 10 Expired
US8552186B2 Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-MET inhibitors Chemistry; Metallurgy 9 Active
US9132128B2 Fused bicyclic 2,4-diaminopyrimidine derivative as a dual ALK and FAK inhibitor Chemistry; Metallurgy 4 Active
US9339502B2 Fused bicyclic 2,4-diaminopyrimidine derivative as a dual ALK and FAK inhibitor Chemistry; Metallurgy 3 Active
US9914730B2 Azaquinazoline inhibitors of Atypical protein Kinase C Chemistry; Metallurgy 3 Active
US9896446B2 Azaquinazoline inhibitors of atypical protein kinase C Chemistry; Metallurgy 2 Active
US9623026B2 Fused bicyclic 2,4-diaminopyrimidine derivative as a dual ALK and FAK inhibitor Chemistry; Metallurgy 2 Active
US11020396B2 Pyrimidinone derivatives as Cdc7 inhibitors Chemistry; Metallurgy 1 Active
US10111872B2 Fused bicyclic 2,4-diaminopyrimidine derivative as a dual ALK and FAK inhibitor Chemistry; Metallurgy 1 Active
US8471005B2 Pyrrolotriazines as ALK and JAK2 inhibitors Human Necessities 1 Active
US9487529B2 Macrocyclic compounds as ALK, FAK and JAK2 inhibitors Chemistry; Metallurgy 1 Active
US10632119B2 Fused bicyclic 2,4-diaminopyrimidine derivative as a dual ALK and FAK inhibitor Chemistry; Metallurgy 0 Active
US9238656B2 Imidazo[4,5-b]pyridine derivatives as ALK and JAK modulators for the treatment of proliferative disorders Chemistry; Metallurgy 0 Active
US12227521B2 CGRP antagonist compounds Chemistry; Metallurgy 0 Active
US9440984B2 Pyrrolotriazines as ALK inhibitors Human Necessities 0 Active
US10919896B2 Preparation and uses of pyrimidinone derivatives Chemistry; Metallurgy 0 Active
US6720329B2 Spiro-cyclic &bgr;-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-&agr; converting enzyme (TACE) Chemistry; Metallurgy 0 Expired
US6962938B2 Spiro-cyclic β-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-α converting enzyme (TACE) Chemistry; Metallurgy 0 Expired
US10954251B2 Thienopyrimidine inhibitors of atypical protein kinase C Chemistry; Metallurgy 0 Active
US11766434B2 Pyrimidinone derivatives as CDC7 inhibitors Chemistry; Metallurgy 0 Active
US12344621B2 CGRP antagonist compounds Chemistry; Metallurgy 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.