Inventor · Ebreichsdorf, AT

Harald Engelhardt

24Patents
8h-index
49Co-inventors
71Inventor score

Filing activity: May 18, 2005 → Oct 29, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US7241769B2 Pyrimidines as PLK inhibitors Chemistry; Metallurgy 60 Expired
US7371753B2 Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions Human Necessities 48 Expired
US10328074B2 Substituted [1,2,4]triazolo[4,3-a]pyrazines as BRD4 inhibitors Chemistry; Metallurgy 26 Active
US7521457B2 Pyrimidines as PLK inhibitors Chemistry; Metallurgy 18 Expired
US7569561B2 2,4-diaminopyrimidines useful for treating cell proliferation diseases Chemistry; Metallurgy 11 Active
US8258129B2 4-heterocycloalkylpyri(mi)dines, process for the preparation thereof and their use as medicaments Chemistry; Metallurgy 9 Active
US8895581B2 1H-imidazo[4,5-c]quinolines Human Necessities 9 Active
US8207179B2 Substituted indolines as tyrosine kinase inhibitors Chemistry; Metallurgy 8 Active
US8575203B2 Chemical compounds Chemistry; Metallurgy 7 Active
US9199988B2 Dihydroquinazolinone analogues Chemistry; Metallurgy 3 Active
US9266891B2 Substituted [1,2,4]triazolo[4,3-A]pyrazines that are BRD4 inhibitors Chemistry; Metallurgy 2 Active
US9102684B2 Indolinone analogues Chemistry; Metallurgy 2 Active
US8637549B2 Pyridons as PDK1 inhibitors Chemistry; Metallurgy 2 Active
US9428515B2 Benzimidazole derivatives Human Necessities 2 Active
US9296748B2 Pyridinones Chemistry; Metallurgy 2 Active
US9428513B2 Triazolopyrazine Chemistry; Metallurgy 2 Active
US9422290B2 Triazolopyridazine Human Necessities 2 Active
US11174245B2 Benzimidazole compounds and derivatives as EGFR inhibitors Chemistry; Metallurgy 0 Active
US11608343B2 Substituted pyrimido[5,4-d]pyrimidines as HER2 inhibitors Chemistry; Metallurgy 0 Active
US11077107B2 Triazolopyrazine Chemistry; Metallurgy 0 Active
US12064421B2 Substituted 1H-pyrazolo[4,3-c]pyridines and derivatives as EGFR inhibitors Human Necessities 0 Active
US11261184B2 [1,6]naphthyridine compounds and derivatives as CDK8/CDK19 inhibitors Human Necessities 0 Active
US11213520B2 Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors Chemistry; Metallurgy 0 Active
US8404674B2 Substituted 9H-purin-2-YL compounds, compositions thereof and uses thereof Human Necessities 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.