Inventor · Vosselaar, BE

Jan Heeres

124Patents
23h-index
85Co-inventors
93Inventor score

Filing activity: Nov 19, 1974 → Jul 2, 2019

Most-cited inventions

PatentTitleAreaCited byStatus
US7514445B2 Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors) Chemistry; Metallurgy 112 Expired
US6197779A HIV inhibiting pyrimidine derivative Chemistry; Metallurgy 111 Expired
US7125879B2 HIV inhibiting pyrimidines derivatives Chemistry; Metallurgy 76 Expired
US4079062A Triazole derivatives Chemistry; Metallurgy 73 Expired
US4267179A Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidaz oles and 1H-1,2,4-triazoles Chemistry; Metallurgy 56 Expired
US7531548B2 HIV inhibiting 5-carbo- or heterocyclic substituted pyrimidines Chemistry; Metallurgy 55 Expired
US4144346A Novel 1-(1,3-dioxolan-2-ylmethyl)-1H-imidazoles Chemistry; Metallurgy 54 Expired
US6440986B2 HIV Inhibiting pyrimidine derivatives Chemistry; Metallurgy 50 Expired
US4791111A [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]- 1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties Chemistry; Metallurgy 44 Expired
US4598085A Fungicidal 1-(2-aryl-2-R-ethyl)-1H-1,2,4-triazoles Chemistry; Metallurgy 40 Expired
US4160838A Antimicrobial and plant-growth-regulating triazole derivatives Chemistry; Metallurgy 38 Expired
US4931444A 5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols Chemistry; Metallurgy 31 Expired
US6150360A Trisubstituted 1,3,5-Triazine Derivatives Chemistry; Metallurgy 31 Expired
US5637592A Acyl derivatives of azolones Chemistry; Metallurgy 27 Expired
US7276510B2 HIV replication inhibitors Chemistry; Metallurgy 26 Expired
US5728700A Sulfonamide compounds of azolones anti-helicobacter agents Chemistry; Metallurgy 26 Expired
US5639754A Urea and thiourea derivatives of azolones Chemistry; Metallurgy 26 Expired
US7923554B2 HIV inhibiting 1,2,4-triazin-6-one derivatives Human Necessities 26 Active
US6878717B2 HIV replication inhibiting pyrimidines Human Necessities 24 Expired
US3936470A 1,3-Dioxolan-2-ylmethylimidazoles Chemistry; Metallurgy 23 Expired
US4916134A 4-[4-[4-[4-[[2-(2,4-difluoro phenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]ph enyl]triazolones Chemistry; Metallurgy 23 Expired
US4223036A 1-(1,3-Dioxolan-2-ylmethyl)-1H-1,2,4-triazoles Chemistry; Metallurgy 23 Expired
US7037917B2 HIV replication inhibiting pyrimidines Human Necessities 23 Expired
US5811426A Urea and thiourea derivatives of azolones Chemistry; Metallurgy 20 Expired
US5571811A Sulfonamide derivatives of azolones Chemistry; Metallurgy 20 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.