Inventor · Saint Louis, MO, US

Michael L. Vazquez

150Patents
21h-index
113Co-inventors
93Inventor score

Filing activity: Oct 21, 1987 → Oct 26, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US4918064A Phenyl glycines for use in reducing neurotoxic injury Chemistry; Metallurgy 56 Expired
US6248775A .alpha.- and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 56 Expired
US6423713B1 Substituted pyrazoles as p38 kinase inhibitors Chemistry; Metallurgy 45 Expired
US6060476A .alpha.- and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 43 Expired
US5843946A .alpha.-and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 43 Expired
US6514977B1 Substituted pyrazoles as p38 kinase inhibitors Chemistry; Metallurgy 41 Expired
US6979686B1 Substituted pyrazoles as p38 kinase inhibitors Chemistry; Metallurgy 41 Expired
US5965588A Sulfonylalkanoylamino hydroxyethylamimo sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 38 Expired
US5521219A Sulfonylalkanoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 35 Expired
US5744481A .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 34 Expired
US5216003A Diacid-containing benzimidazole compounds for treatment of neurotoxic injury Chemistry; Metallurgy 33 Expired
US5830897A .alpha.- and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Human Necessities 29 Expired
US6617324B1 Substituted pyrazoles as p38 kinase inhibitors Chemistry; Metallurgy 28 Expired
US5968942A .alpha.- and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 27 Expired
US5508294A Sulfonylalkanoylamino hydroxyethlamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 24 Expired
US6046190A Hydroxyethylamino sulphonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 23 Expired
US6143892A Process for making 5-substituted pyrazoles Chemistry; Metallurgy 23 Expired
US6525059B1 Substituted pyrazoles as p38 kinase inhibitors Chemistry; Metallurgy 23 Expired
US5760064A Sulfonylalkanoylamino hydroxyethylamino sulfanamides useful as retroviral protease inhibitors Chemistry; Metallurgy 23 Expired
US5463104A Succinoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 21 Expired
US5714605A Succinoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 21 Expired
US5639769A Sulfonylalkanoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 20 Expired
US5482947A Retroviral protease inhibitors Chemistry; Metallurgy 20 Expired
US5786483A .alpha.-and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors Chemistry; Metallurgy 19 Expired
US5648511A Method for making intermediates useful in the synthesis of retroviral protease inhibitors Chemistry; Metallurgy 19 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.