Inventor · Basel, CH

Pascal Furet

97Patents
15h-index
190Co-inventors
87Inventor score

Filing activity: May 3, 1993 → Mar 15, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US5981533A Pyrazole derivatives and processes for the preparation thereof Human Necessities 89 Expired
US7083983B2 Inhibitors of the interaction between P53 and MDM2 Chemistry; Metallurgy 79 Expired
US8552002B2 Compounds and compositions as protein kinase inhibitors Chemistry; Metallurgy 77 Active
US7667039B2 1,3-dihydro-imidazo [4,5-C] quinolin-2-ones as lipid kinase inhibitors Human Necessities 62 Active
US7169791B2 Inhibitors of tyrosine kinases Chemistry; Metallurgy 60 Expired
US5686457A Pyrrolopyrimidine derivatives having pharmacological activity Human Necessities 60 Expired
US7122547B1 Anthranilic acid amides and the use thereof as medicaments Human Necessities 57 Expired
US7795273B2 Pyrazolo[1,5-a]pyridine-3-carboxylic acids as EphB and VEGFR2 kinase inhibitors Human Necessities 45 Active
US8815901B2 Quinoline carboxamide derivatives as protein tyrosine kinase inhibitors Chemistry; Metallurgy 39 Active
US8026247B2 Bicyclic amides as kinase inhibitors Chemistry; Metallurgy 36 Active
US6878720B2 VEGF receptor tyrosine kinase inhibitors Chemistry; Metallurgy 25 Expired
US6448277B2 VEGF receptor tyrosine kinase inhibitors Chemistry; Metallurgy 24 Expired
US6096749A Pyrrolopyrimidine derivatives having pharmacological activity Human Necessities 22 Expired
US5683997A Substituted benzazepinones Human Necessities 15 Expired
US9266883B2 Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors Chemistry; Metallurgy 15 Active
US7189729B2 Methods and compositions as protein kinase inhibitors Chemistry; Metallurgy 15 Expired
US7326699B2 4-Amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3-d)pyrimidine derivatives Human Necessities 15 Expired
US5332729A N-aralkyl- and N-heteroaralkyl-aminoalkanephosphinic acids Chemistry; Metallurgy 14 Expired
US8440693B2 Substituted isoquinolinones and quinazolinones Chemistry; Metallurgy 13 Active
US7652022B2 Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases Chemistry; Metallurgy 13 Expired
US8431592B2 1,3-dihydro-imidazo[4,5-c]quinolin-2-ones as lipid kinase inhibitors Human Necessities 12 Active
US8293746B2 Pyrimidinyl aryl urea derivatives being FGF inhibitors Chemistry; Metallurgy 12 Active
US9533988B2 Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors Chemistry; Metallurgy 12 Active
US7002022B2 N-Aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF Chemistry; Metallurgy 10 Expired
US7994170B2 1,3-dihydro-imidazo[4,5-C]quinolin-2-ones as lipid kinase inhibitors Human Necessities 9 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.