Robert W. DeSimone
34Patents
15h-index
40Co-inventors
77Inventor score
Filing activity: Jun 5, 1995 → May 17, 2006
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US6723730B2 | Capsaicin receptor ligands | Chemistry; Metallurgy | 75 | Expired |
| US7160885B2 | Certain 6, 8-(heteroaryl or aryl) disubstituted imidazo[1,2-a]pyrazines as modulators of Hsp90 complex activity | Human Necessities | 59 | Expired |
| US6271241A | Cycloalkyl and aryl fused aminoalkyl-imidazole derivatives: modulators and GLP-1 receptors | Physics | 52 | Expired |
| US7405295B2 | Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds | Human Necessities | 50 | Expired |
| US7312341B2 | 6-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereof | Human Necessities | 44 | Expired |
| US7189723B2 | Certain 8-heteroaryl-6-phenyl-imidazo[1,2-a]pyrazines as modulators of kinase activity | Human Necessities | 43 | Expired |
| US7259164B2 | Certain substituted imidazo[1,2-a]pyrazines, as modulators of kinase activity | Human Necessities | 41 | Expired |
| US6919340B2 | Imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereof | Human Necessities | 41 | Expired |
| US7393848B2 | Certain heterocyclic substituted imidazo[1,2-A]pyrazin-8-ylamines and methods of inhibition of Bruton's tyrosine kinase by such compounds | Chemistry; Metallurgy | 34 | Expired |
| US6380210B1 | Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors | Chemistry; Metallurgy | 27 | Expired |
| US6133265A | Certain amido- and amino- substituted benzylamine derivatives; a new class of neuropeptide Y1 specific ligands | Chemistry; Metallurgy | 27 | Expired |
| US7160879B2 | Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1H-benzoimidazole analogues | Chemistry; Metallurgy | 21 | Expired |
| US7015227B2 | Certain amino-substituted monocycles as kinase modulators | Chemistry; Metallurgy | 16 | Expired |
| US6399604B1 | Substituted 4-OXO-napthyridine-3-carboxamides; GABA brain receptor ligands | Chemistry; Metallurgy | 16 | Expired |
| US6143760A | Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands | Chemistry; Metallurgy | 16 | Expired |
| US6316617A | Certain amido-and amino-substituted benzylamine derivatives; a new class of Neuropeptide Y1 specific ligands | Chemistry; Metallurgy | 15 | Expired |
| US6646124B2 | Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands | Chemistry; Metallurgy | 12 | Expired |
| US5637724A | Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands | Chemistry; Metallurgy | 8 | Expired |
| US6358949B1 | Aryl and hetroaryl fused aminoalkyl-imidazole derivatives: selective modulators of bradykinin B2 receptors | Chemistry; Metallurgy | 7 | Expired |
| US5637725A | Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands | Chemistry; Metallurgy | 5 | Expired |
| US6127395A | Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands | Chemistry; Metallurgy | 5 | Expired |
| US5936095A | Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands | Chemistry; Metallurgy | 4 | Expired |
| US6509366B2 | Substituted imidazoles as selective modulators of Bradykinin B2 receptors | Chemistry; Metallurgy | 4 | Expired |
| US6627624B1 | Aryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors | Chemistry; Metallurgy | 3 | Expired |
| US5849927A | Substituted aryl and cycloalkyl imidazolones; a new class of GABA brain receptor ligands | Chemistry; Metallurgy | 3 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.