Inventor · Waltham, MA, US

Ruoxi Lan

37Patents
7h-index
46Co-inventors
69Inventor score

Filing activity: Oct 4, 2000 → Aug 13, 2020

Most-cited inventions

PatentTitleAreaCited byStatus
US9969710B2 Heteroaryl compounds as IRAK inhibitors and uses thereof Emerging Cross-Sectional Technologies 32 Active
US7452862B2 Conformationally-controlled biologically active macrocyclic small molecules as motilin antagonists or ghrelin agonists Chemistry; Metallurgy 13 Expired
US7169899B1 Combinatorial synthesis of libraries of macrocyclic compounds useful in drug discovery Emerging Cross-Sectional Technologies 12 Expired
US8637532B2 Amino azaheterocyclic carboxamides Chemistry; Metallurgy 9 Active
US8569295B2 Bicyclic urea compounds Chemistry; Metallurgy 7 Active
US9624246B2 Pyridazinone macrocycles as IRAK inhibitors and uses thereof Chemistry; Metallurgy 7 Active
US9708324B2 Macrocyclic compounds as IRAK1/4 inhibitors and uses thereof Chemistry; Metallurgy 7 Active
US9815836B2 Macrocyclic compounds as IRAK1/4 inhibitors and uses thereof Chemistry; Metallurgy 6 Active
US9580443B2 Heterocyclic derivatives as modulators of kinase activity Human Necessities 5 Active
US8008440B2 Combinatorial synthesis of libraries of macrocyclic compounds useful in drug discovery Emerging Cross-Sectional Technologies 5 Active
US9440968B2 Substituted pyrido[3,2-d]pyrimidines for treating cancer Chemistry; Metallurgy 5 Active
US9145392B2 Imidazole amines as modulators of kinase activity Chemistry; Metallurgy 4 Active
US8022252B2 Spatially-defined macrocyclic compounds useful for drug discovery Chemistry; Metallurgy 3 Active
US9139568B2 Heterocyclic carboxamides as modulators of kinase activity Chemistry; Metallurgy 3 Active
US9321760B2 Aminopyrimidine derivatives for use as modulators of kinase activity Chemistry; Metallurgy 2 Active
US10836750B1 TLR7/8 antagonists and uses thereof Chemistry; Metallurgy 2 Active
US10793553B2 TLR7/8 antagonists and uses thereof Chemistry; Metallurgy 2 Active
US9458134B2 Heterocycles as modulators of kinase activity Chemistry; Metallurgy 2 Active
US9040560B2 Amino azaheterocyclic carboxamides Chemistry; Metallurgy 2 Active
US8710044B2 Bicyclic azaheterocyclic carboxamides Chemistry; Metallurgy 1 Active
US9018419B2 Combinatorial synthesis of libraries of macrocyclic compounds useful in drug discovery Emerging Cross-Sectional Technologies 1 Active
US10517872B2 Pyridazinone macrocycles as IRAK inhibitors and uses thereof Chemistry; Metallurgy 1 Active
US9662330B2 Aminopyrimidine derivatives for use as modulators of kinase activity Chemistry; Metallurgy 1 Active
US9434714B2 Pyrimidine imidazole amines as modulators of kinase activity Human Necessities 1 Active
US10080750B2 Aminopyrimidine derivatives for use as modulators of kinase activity Chemistry; Metallurgy 1 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.