Inventor · East Haven, CT, US

Scott A. Mitchell

67Patents
19h-index
113Co-inventors
87Inventor score

Filing activity: Jul 12, 2002 → Dec 18, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US7160885B2 Certain 6, 8-(heteroaryl or aryl) disubstituted imidazo[1,2-a]pyrazines as modulators of Hsp90 complex activity Human Necessities 59 Expired
US7405295B2 Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds Human Necessities 50 Expired
US8450321B2 6-(1H-indazol-6-yl)-N-[4-(morpholin-4-yl)phenyl]imidazo-[1,2-A]pyrazin-8-amine, or a pharmaceutically acceptable salt thereof, as a SYK inhibitor Chemistry; Metallurgy 45 Active
US7312341B2 6-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereof Human Necessities 44 Expired
US7189723B2 Certain 8-heteroaryl-6-phenyl-imidazo[1,2-a]pyrazines as modulators of kinase activity Human Necessities 43 Expired
US7259164B2 Certain substituted imidazo[1,2-a]pyrazines, as modulators of kinase activity Human Necessities 41 Expired
US6919340B2 Imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereof Human Necessities 41 Expired
US8455493B2 Imidazopyrazine Syk inhibitors Physics 36 Active
US8440667B2 Imidazopyrazine Syk inhibitors Physics 34 Active
US7393848B2 Certain heterocyclic substituted imidazo[1,2-A]pyrazin-8-ylamines and methods of inhibition of Bruton's tyrosine kinase by such compounds Chemistry; Metallurgy 34 Expired
US8748607B2 Imidazopyrizine syk inhibitors Physics 30 Active
US8765761B2 6-(1H-indazol-6-yl)-N-{4-[2-methyl-1-(morpholin-4-yl)propan-2-yl]phenyl}imidazo[1,2-A]pyrazin-8-amine, or a pharmaceutically acceptable salt thereof, as a syk inhibitor Physics 29 Active
US8697699B2 Imidazopyrazine SYK inhibitors Human Necessities 27 Active
US8796270B2 N-[6-(1H-indazol-6-yl)imidazo[1,2-A]pyridin-8-yl]-6-(morpholin-4-yl)pyridazin-3-amine, or a pharmaceutically acceptable salt thereof, as a SYK inhibitor Physics 25 Active
US9120811B2 6-(1H-indazol-6-YL)-N-(4-morpholinophenyl)imidazo[1,4-A]pyrazin-8-amine for treating leukemia or lymphoma Physics 25 Active
US7884108B2 Certain substituted pyrazinones Chemistry; Metallurgy 22 Active
US8962835B2 Imidazopyrazine Syk inhibitors Physics 21 Active
US8618107B2 Pyridone and aza-pyridone compounds and methods of use Chemistry; Metallurgy 20 Active
US9212191B2 6-(2,3-dihydro-1H-pyrido-[2,3-b][1,4]oxazin-7-yl)-N-(4-morpholinophenyl)imidazo[1,2-a] pyrazin-8-amine as a spleen tyrosine kinase inhibitor Physics 19 Active
US9290505B2 Substituted imidazo[1,2-a]pyrazines as Syk inhibitors Chemistry; Metallurgy 19 Active
US8058446B2 Certain substituted amides, method of making, and method of use thereof Chemistry; Metallurgy 18 Active
US9504684B2 Syk inhibitors Human Necessities 18 Active
US7015227B2 Certain amino-substituted monocycles as kinase modulators Chemistry; Metallurgy 16 Expired
US7838523B2 Certain substituted amides, method of making, and method of use thereof Chemistry; Metallurgy 16 Active
US9567348B2 Substituted pyrazolo[1,5-a]pyrimidines as Syk inhibitors Physics 15 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.