Chemical modifications of monomers and oligonucleotides with cycloaddition
US8962580B2 · kind B2 · utility
22Cited by
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11Claims
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Key dates
| Filing date | Sep 23, 2009 |
| Grant date | Feb 24, 2015 |
| Priority date | — |
| Expiry date | Jan 7, 2032 |
Classification
- Technology area (CPC Y)Emerging Cross-Sectional Technologies
- CPC primaryY02A50/30
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The invention features compounds of formula I or II:In one embodiment, the invention relates compounds and processes for conjugating ligand to oligonucleotide. The invention further relates to methods for treating various disorders and diseases such as viral infections, bacterial infections, parasitic infections, cancers, allergies, autoimmune diseases, immunodeficiencies and immunosuppression.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.