Inventor · Carlsbad, CA, US

Muthiah Manoharan

322Patents
56h-index
168Co-inventors
93Inventor score

Filing activity: Sep 3, 1993 → Oct 8, 2024

Most-cited inventions

PatentTitleAreaCited byStatus
US5459255A N-2 substituted purines Chemistry; Metallurgy 758 Expired
US5587469A Oligonucleotides containing N-2 substituted purines Chemistry; Metallurgy 574 Expired
US5681941A Substituted purines and oligonucleotide cross-linking Chemistry; Metallurgy 556 Expired
US5578718A Thiol-derivatized nucleosides Chemistry; Metallurgy 341 Expired
US8158601B2 Lipid formulation Emerging Cross-Sectional Technologies 293 Active
US6335434B1 Nucleosidic and non-nucleosidic folate conjugates Chemistry; Metallurgy 287 Expired
US6210892A Alteration of cellular behavior by antisense modulation of mRNA processing Emerging Cross-Sectional Technologies 245 Expired
US9345780B2 Site specific delivery of nucleic acids by combining targeting ligands with endosomolytic components Chemistry; Metallurgy 237 Active
US6528631B1 Oligonucleotide-folate conjugates Chemistry; Metallurgy 231 Expired
US8106022B2 Carbohydrate conjugates as delivery agents for oligonucleotides Emerging Cross-Sectional Technologies 229 Active
US6153737A Derivatized oligonucleotides having improved uptake and other properties Chemistry; Metallurgy 212 Expired
US6147200A 2'-O-acetamido modified monomers and oligomers Chemistry; Metallurgy 190 Expired
US6600032B1 2′-O-aminoethyloxyethyl-modified oligonucleotides Chemistry; Metallurgy 184 Expired
US6300319A Targeted oligonucleotide conjugates Chemistry; Metallurgy 180 Expired
US6656730B1 Oligonucleotides conjugated to protein-binding drugs Chemistry; Metallurgy 176 Expired
US8828956B2 Carbohydrate conjugates as delivery agents for oligonucleotides Emerging Cross-Sectional Technologies 160 Active
US6867294B1 Gapped oligomers having site specific chiral phosphorothioate internucleoside linkages Chemistry; Metallurgy 158 Expired
US6242589A Phosphorothioate oligonucleotides having modified internucleoside linkages Chemistry; Metallurgy 146 Expired
US8450467B2 Carbohydrate conjugates as delivery agents for oligonucleotides Emerging Cross-Sectional Technologies 145 Active
US8642076B2 Lipid containing formulations Human Necessities 138 Active
US6127533A 2'-O-aminooxy-modified oligonucleotides Emerging Cross-Sectional Technologies 129 Expired
US6762169B1 Ligand-conjugated oligomeric compounds Chemistry; Metallurgy 128 Expired
US6395492B1 Derivatized oligonucleotides having improved uptake and other properties Chemistry; Metallurgy 121 Expired
US6271358A RNA targeted 2'-modified oligonucleotides that are conformationally preorganized Chemistry; Metallurgy 119 Expired
US7723509B2 IRNA agents with biocleavable tethers Chemistry; Metallurgy 118 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.