Inventor · Basel, CH

Alexander Alanine

38Patents
9h-index
52Co-inventors
78Inventor score

Filing activity: Jul 14, 1997 → Jul 15, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US6407094B1 Glutamate receptor antagonists Human Necessities 45 Expired
US6509328B1 Glutamate receptor antagonists Chemistry; Metallurgy 33 Expired
US6521754B2 Benzothiazole derivatives with activity as adenosine receptor ligands Chemistry; Metallurgy 26 Expired
US5889026A 4-hydroxy-piperodine derivatives Chemistry; Metallurgy 23 Expired
US6451819B2 Heterocyclic compounds useful as NMDA receptor selective subtype blockers Chemistry; Metallurgy 20 Expired
US6265426A Triazole derivatives Chemistry; Metallurgy 14 Expired
US6963000B2 Benzothiazole derivatives with activity as adenosine receptor ligands Chemistry; Metallurgy 13 Expired
US6339093B1 Isoquinoline derivatives Chemistry; Metallurgy 10 Expired
US6432985B1 Neuroprotective substituted piperidine compounds with activity as NMDA NR2B subtype selective antagonists Human Necessities 9 Expired
US6610723B2 Imidazole derivatives Chemistry; Metallurgy 6 Expired
US6831087B2 Pyridine substituted isoquinoline derivatives Human Necessities 5 Expired
US6440995B1 Quinolin-4-yl derivatives Chemistry; Metallurgy 5 Expired
US6835732B2 Benzothiazole derivatives with activity as adenosine receptor ligands Chemistry; Metallurgy 4 Expired
US7151098B2 Glutamate receptor antagonists Chemistry; Metallurgy 4 Expired
US6184236A Method of treating a neurodegenerative disease by administering an aryl-cyclohexylamine derivative Human Necessities 4 Expired
US6359138B1 4-hydroxy-piperidine derivatives Chemistry; Metallurgy 4 Expired
US6310213A Ethanesulfonyl-piperidine derivatives Chemistry; Metallurgy 4 Expired
US6407235B1 Prodrug acid esters of [2-(4-benzyl-3-hydroxy-piperidin-1-yl)-ethansulfonyl]phenol Chemistry; Metallurgy 3 Expired
US11098080B2 Peptide macrocycles against Acinetobacter baumannii Emerging Cross-Sectional Technologies 3 Active
US11066443B2 Anti-bacterial peptide macrocycles and use thereof Emerging Cross-Sectional Technologies 3 Active
US6071929A Octahydro phenanthridine derivatives useful as NMDA-R receptor subtype blockers Chemistry; Metallurgy 3 Expired
US6960578B2 Glutamate receptor antagonists Chemistry; Metallurgy 3 Expired
US6015824A Pyrrolidine and piperidine derivatives and treatment of neurodegenerative disorders Human Necessities 3 Expired
US5952344A Tetrahydroisoquinoline derivatives Chemistry; Metallurgy 3 Expired
US7317007B2 Benzothiazole derivatives with activity as adenosine receptor ligands Chemistry; Metallurgy 2 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.