Inventor · Hilden, DE

Alexandros Vakalopoulos

53Patents
8h-index
99Co-inventors
77Inventor score

Filing activity: Dec 15, 2005 → Aug 11, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US9023849B2 Substituted fused imidazoles and pyrazoles and use thereof Chemistry; Metallurgy 26 Active
US8426602B2 Heteroaryl-substituted dicyanopyridines and their use Chemistry; Metallurgy 24 Active
US8859569B2 Substituted annellated pyrimidines and use thereof Chemistry; Metallurgy 24 Active
US9126998B2 Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use Human Necessities 11 Active
US8778964B2 Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use Human Necessities 11 Active
US8796305B2 Carboxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use Chemistry; Metallurgy 10 Active
US8946215B2 Hydroxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use Human Necessities 9 Active
US8673903B2 Substituted 8-alkoxy-2-aminotetralin derivatives, and use thereof Chemistry; Metallurgy 9 Active
US8420825B2 Alkylamino-substituted dicyanopyridines and their amino acid ester prodrugs Chemistry; Metallurgy 6 Active
US8440700B2 Substituted aryloxazoles and their use Chemistry; Metallurgy 5 Active
US9266871B2 Trifluoromethyl-substituted fused pyrimidines and their use Chemistry; Metallurgy 5 Active
US10435403B2 Positive allosteric modulators of muscarinic M2 receptor Chemistry; Metallurgy 5 Active
US8304412B2 Cyclically substituted 3,5-dicyano-2-thiopyridines and use thereof Chemistry; Metallurgy 4 Active
US9422285B2 Substituted pyrazolo[1,5-A]-pyridine-3-carboxamides and use thereof Chemistry; Metallurgy 4 Active
US9776997B2 3-aryl-substituted imidazo[1,2-A]pyridines and their use Human Necessities 3 Active
US9605008B2 Benzyl-1H-pyrazolo[3,4-b]pyridines and use thereof Human Necessities 3 Active
US9498480B2 Substituted azabicycles and use thereof Chemistry; Metallurgy 3 Active
US9624214B2 Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use Chemistry; Metallurgy 2 Active
US10150773B2 N-substituted 8-[(2,6-difluorobenzyl)oxy]-2,6- dimethylimidazo[1,2-a]pyrazin-3-carboxamide derivatives as stimulators of soluble guanylate cyclase (SGC) for the treatment of cardiovascular diseases Chemistry; Metallurgy 2 Active
US9387203B2 Substituted aminoindane- and aminotetralinecarboxylic acids and the use thereof Chemistry; Metallurgy 2 Active
US8772498B2 Alkylamine-substituted dicyanopyridine and amino acid ester prodrugs thereof Chemistry; Metallurgy 2 Active
US10519154B2 7-substituted 1-pyridyl-naphthyridine-3-carboxylic acid amides and use thereof Chemistry; Metallurgy 2 Active
US9688699B2 3-(pyrimidine-2-yl)imidazo[1,2-a]pyridines Human Necessities 1 Active
US8741834B2 Dipeptoid prodrugs and the use thereof Chemistry; Metallurgy 1 Active
US8227511B2 Substituted chromanol derivatives and their use Chemistry; Metallurgy 1 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.