Inventor · Chelmsford, GB

Angus Murray MacLeod

82Patents
14h-index
94Co-inventors
87Inventor score

Filing activity: Mar 19, 1987 → Aug 16, 2022

Most-cited inventions

PatentTitleAreaCited byStatus
US5514718A Heterocyclic compounds, processes for their preparation and pharmaceutical compositions containing them Chemistry; Metallurgy 531 Expired
US5334606A Oxazolidindione substituted indole derivatives Chemistry; Metallurgy 52 Expired
US5885999A Serine derivatives and their use as therapeutic agents Chemistry; Metallurgy 45 Expired
US5612337A Substituted morpholine derivatives and their use as therapeutic agents Chemistry; Metallurgy 38 Expired
US5620989A 4-Arylmethyloxymethyl piperidines as tachykinin antagonsits Chemistry; Metallurgy 33 Expired
US6136824A 1-piperidinyl-propan-2-derivatives and their use as therapeutic agents Chemistry; Metallurgy 30 Expired
US5760018A Gem-disubstituted azacyclic tachykinin antagonists Chemistry; Metallurgy 30 Expired
US6200975A Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligands Human Necessities 18 Expired
US5242927A Prodrugs for oxadiazole muscarinic agonists Chemistry; Metallurgy 17 Expired
US5472978A Aromatic compounds, pharmaceutical compositions containing them and their use in therapy Chemistry; Metallurgy 15 Expired
US5849746A Substituted 1,4-piperazine-heteroaryl derivatives as 5-HT.sub.1D receptor agonists Human Necessities 15 Expired
US5519163A Inhibitors of phosphoinositide-specific phospholipase C Chemistry; Metallurgy 14 Expired
US5405853A Thiadiazoles useful in the treatment of senile dementia Chemistry; Metallurgy 14 Expired
US5973156A Piperidine and tetrahydropyridine derivatives Chemistry; Metallurgy 14 Expired
US5661162A 4-aminomethyl/thiomethyl/sulfonylmethyl-4-phenylpiperdines as tachykinin receptor antagonists Chemistry; Metallurgy 13 Expired
US7381725B2 Pyridazine derivatives as ligands for GABA receptors Chemistry; Metallurgy 12 Expired
US6211219A Aminocyclohexane derivatives as 5-HT receptor agonists Chemistry; Metallurgy 12 Expired
US5977116A Piperazine, piperidine and tetrahydropyridine derivatives Chemistry; Metallurgy 10 Expired
US7501411B2 Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases Human Necessities 10 Active
US5328927A Hetercyclic compounds, processes for their preparation and pharmaceutical compositions containing them Chemistry; Metallurgy 9 Expired
US6310203A Precursor compounds to substituted 1,2,4-triazolo[3,4,-a]phathalazine GABA alpha 5 ligands Human Necessities 9 Expired
US5998440A Azetidine, pyrrolidine and piperidine derivatives Chemistry; Metallurgy 8 Expired
US7915256B2 Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases Human Necessities 7 Active
US6127388A Azetidine, pyrrolidine and piperidine derivatives as 5-HT.sub.1D receptor agonists Human Necessities 6 Expired
US7030128B2 Imidazo-pyrimidine derivatives as ligands for GABA receptors Human Necessities 6 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.