Angus Murray MacLeod
82Patents
14h-index
94Co-inventors
87Inventor score
Filing activity: Mar 19, 1987 → Aug 16, 2022
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US5514718A | Heterocyclic compounds, processes for their preparation and pharmaceutical compositions containing them | Chemistry; Metallurgy | 531 | Expired |
| US5334606A | Oxazolidindione substituted indole derivatives | Chemistry; Metallurgy | 52 | Expired |
| US5885999A | Serine derivatives and their use as therapeutic agents | Chemistry; Metallurgy | 45 | Expired |
| US5612337A | Substituted morpholine derivatives and their use as therapeutic agents | Chemistry; Metallurgy | 38 | Expired |
| US5620989A | 4-Arylmethyloxymethyl piperidines as tachykinin antagonsits | Chemistry; Metallurgy | 33 | Expired |
| US6136824A | 1-piperidinyl-propan-2-derivatives and their use as therapeutic agents | Chemistry; Metallurgy | 30 | Expired |
| US5760018A | Gem-disubstituted azacyclic tachykinin antagonists | Chemistry; Metallurgy | 30 | Expired |
| US6200975A | Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligands | Human Necessities | 18 | Expired |
| US5242927A | Prodrugs for oxadiazole muscarinic agonists | Chemistry; Metallurgy | 17 | Expired |
| US5472978A | Aromatic compounds, pharmaceutical compositions containing them and their use in therapy | Chemistry; Metallurgy | 15 | Expired |
| US5849746A | Substituted 1,4-piperazine-heteroaryl derivatives as 5-HT.sub.1D receptor agonists | Human Necessities | 15 | Expired |
| US5519163A | Inhibitors of phosphoinositide-specific phospholipase C | Chemistry; Metallurgy | 14 | Expired |
| US5405853A | Thiadiazoles useful in the treatment of senile dementia | Chemistry; Metallurgy | 14 | Expired |
| US5973156A | Piperidine and tetrahydropyridine derivatives | Chemistry; Metallurgy | 14 | Expired |
| US5661162A | 4-aminomethyl/thiomethyl/sulfonylmethyl-4-phenylpiperdines as tachykinin receptor antagonists | Chemistry; Metallurgy | 13 | Expired |
| US7381725B2 | Pyridazine derivatives as ligands for GABA receptors | Chemistry; Metallurgy | 12 | Expired |
| US6211219A | Aminocyclohexane derivatives as 5-HT receptor agonists | Chemistry; Metallurgy | 12 | Expired |
| US5977116A | Piperazine, piperidine and tetrahydropyridine derivatives | Chemistry; Metallurgy | 10 | Expired |
| US7501411B2 | Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases | Human Necessities | 10 | Active |
| US5328927A | Hetercyclic compounds, processes for their preparation and pharmaceutical compositions containing them | Chemistry; Metallurgy | 9 | Expired |
| US6310203A | Precursor compounds to substituted 1,2,4-triazolo[3,4,-a]phathalazine GABA alpha 5 ligands | Human Necessities | 9 | Expired |
| US5998440A | Azetidine, pyrrolidine and piperidine derivatives | Chemistry; Metallurgy | 8 | Expired |
| US7915256B2 | Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases | Human Necessities | 7 | Active |
| US6127388A | Azetidine, pyrrolidine and piperidine derivatives as 5-HT.sub.1D receptor agonists | Human Necessities | 6 | Expired |
| US7030128B2 | Imidazo-pyrimidine derivatives as ligands for GABA receptors | Human Necessities | 6 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.