Anthony Marfat
62Patents
15h-index
44Co-inventors
84Inventor score
Filing activity: May 2, 1984 → Jan 27, 2022
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US5814651A | Catechol diethers as selective PDE.sup.IV inhibitors | Chemistry; Metallurgy | 71 | Expired |
| US5059609A | Substituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseases | Emerging Cross-Sectional Technologies | 60 | Expired |
| US5322847A | Azabenzimidazoles in the treatment of asthma, arthritis and related diseases | Chemistry; Metallurgy | 55 | Expired |
| US6380218B1 | Nicotinamide derivatives | Chemistry; Metallurgy | 54 | Expired |
| US6740655B2 | Pyrimidine carboxamides useful as inhibitors of PDE4 isozymes | Chemistry; Metallurgy | 52 | Expired |
| US6559168B2 | Thiazolyl-acid amide derivatives useful as inhibitors of PDE4 isozymes | Chemistry; Metallurgy | 38 | Expired |
| US5998451A | Substituted tetralins, chromans and related compounds in the treatment and related compounds in the treatment of asthma, arthritis and related diseases | Emerging Cross-Sectional Technologies | 24 | Expired |
| US6391872B1 | Indazole bioisostere replacement of catechol in therapeutically active compounds | Human Necessities | 23 | Expired |
| US6649633B2 | Nicotinamide biaryl derivatives useful as inhibitors of PDE4 isozymes | Chemistry; Metallurgy | 21 | Expired |
| US5116854A | Anti-inflammatory 1-heteroaryl-3-acyl-2-oxindoles | Chemistry; Metallurgy | 19 | Expired |
| US6716978B2 | Therapeutically active compounds based on indazole bioisostere replacement of catechol in PDE4 inhibitors | Emerging Cross-Sectional Technologies | 19 | Expired |
| US5811432A | Azaoxindole derivatives | Chemistry; Metallurgy | 17 | Expired |
| US6262040A | Indazole derivatives and their use as inhibitors of phosphodiesterase (PDE) type IV and the production of tumor necrosis factor (TNF) | Chemistry; Metallurgy | 16 | Expired |
| US5958953A | Substituted indazole derivatives | Chemistry; Metallurgy | 16 | Expired |
| US4551452A | Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor | Chemistry; Metallurgy | 15 | Expired |
| US6040329A | Substituted indazole analogs | Human Necessities | 10 | Expired |
| US7354941B2 | Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of PDE4 isozymes | Chemistry; Metallurgy | 10 | Expired |
| US5384318A | Substituted sulfonamides and related compounds in the treatment of asthma, arthritis and related diseases | Chemistry; Metallurgy | 9 | Expired |
| US5298512A | Substituted chromans and their use in the treatment of asthma, arthritis and related diseases | Chemistry; Metallurgy | 7 | Expired |
| US6166031A | Substituted tetralins, chromans and related compounds in the treatment of asthma | Human Necessities | 7 | Expired |
| US5698550A | Tetralin and chroman derivatives useful in the treatment of asthma, arthritis and related diseases | Chemistry; Metallurgy | 6 | Expired |
| US9988394B2 | Oxabicycloheptane prodrugs | Chemistry; Metallurgy | 6 | Active |
| US7250518B2 | Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes | Chemistry; Metallurgy | 6 | Expired |
| US8901105B2 | Prodrug derivatives of (E)-N-methyl-N-((3-M ethylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide | Human Necessities | 6 | Active |
| US10364252B2 | Oxabicycloheptane prodrugs | Chemistry; Metallurgy | 6 | Active |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.