Inventor · Budapest, HU

Gyula Simig

54Patents
5h-index
219Co-inventors
75Inventor score

Filing activity: Sep 11, 1981 → Feb 16, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US6469168B1 Piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for the preparation of the active substance Human Necessities 42 Expired
US6046337A Process for the preparation of a dihydropyridine derivative Chemistry; Metallurgy 16 Expired
US7951798B2 Polymorphs of olanzapine hydrochloride Human Necessities 6 Active
US6646133B1 Process for the preparation of amorphous atorvastatin calcium Chemistry; Metallurgy 6 Expired
US4559406A Process for the preparation of aminolactone carboxylic acid Emerging Cross-Sectional Technologies 5 Expired
US4665083A Iminothiazolidine derivatives Human Necessities 5 Expired
US7060842B2 Method for synthesis of (2S, 3aS, 7aS)-1-{(S)-alanyl}-octahydro-1H -indole-2-carboxylic acid derivatives and use for synthesis of perindopril Emerging Cross-Sectional Technologies 4 Expired
US5523303A Trisubstituted cycloalkane derivatives and process for the preparation thereof Chemistry; Metallurgy 3 Expired
US5652270A Pharmaceutical compositions containing bicycloheptane ether amines and a process for the preparation thereof Human Necessities 3 Expired
US6242386A Process for preparing (1R,2S,4R)-(-)-2-[(2'-{N,N-dimethylamino}-ethoxy)]-2-[phenyl]-1,7,7-tri-[m ethyl]-bicyclo[2.2.1]heptane and pharmaceutically acceptable acid addition salts thereof Chemistry; Metallurgy 3 Expired
US5912245A Acid amide derivatives and process for the preparation thereof Human Necessities 3 Expired
US7183283B2 Piperidinyl-alkylamino-pyridazinone derivatives, a process for the preparation thereof and pharmaceutical compositions containing said compounds Human Necessities 3 Expired
US6130215A Piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same and a process for the preparation of the novel compounds Chemistry; Metallurgy 3 Expired
US6930110B2 Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same Chemistry; Metallurgy 2 Expired
US6335469B1 High purity (1R,2S,4R)-(-)-2-[(2′-{N,N-dimethylamino}-ethoxy)]-2-[phenyl]-1,7,7-tri-[methyl]-bicyclo[2.2.1]heptane and pharmaceutically acceptable acid addition salts thereof Chemistry; Metallurgy 2 Expired
US7851627B2 Optically active carbamates, process for preparation thereof and use thereof as pharmaceutical intermediates Chemistry; Metallurgy 2 Active
US5486528A Basic ethers and process for the preparation thereof Chemistry; Metallurgy 2 Expired
US4435322A Heterocyclic compounds containing an alkoxycarbonyl and a substituted methyl group Fixed Constructions 1 Expired
US7910591B2 Piperazine derivatives of alkyl oxindoles Chemistry; Metallurgy 1 Expired
US8507513B2 Process for the preparation of rosuvastatin salts Human Necessities 1 Active
US5545741A Process for the preparation of epibatidine Human Necessities 1 Expired
US7307168B2 Process for the preparation of 3-{2-′4- (6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyllethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido′1,2-methyl-4h-pyrido′,2-a!pyrimidin-4-one Chemistry; Metallurgy 1 Expired
US7189711B2 2, 3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient Human Necessities 1 Expired
US5716986A Oxaindene derivatives and process for the preparation thereof Chemistry; Metallurgy 1 Expired
US4432901A Beta-lactam compounds containing a C-acetal group and process for their preparation Emerging Cross-Sectional Technologies 1 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.