Marcus Koppitz
26Patents
5h-index
82Co-inventors
72Inventor score
Filing activity: Apr 8, 1999 → Aug 21, 2020
Most-cited inventions
| Patent | Title | Area | Cited by | Status |
|---|---|---|---|---|
| US9549932B2 | 2-(morpholin-4-yl)-1,7-naphthyridines | Chemistry; Metallurgy | 16 | Active |
| US7122570B2 | Tetrahydrocarbazol derivatives as ligands for G-protein-coupled receptors (GPCR) | Human Necessities | 11 | Expired |
| US9340528B2 | Substituted aminoquinoxalines as tyrosine threonine kinase inhibitors | Chemistry; Metallurgy | 10 | Active |
| US10729680B2 | 5-substituted 2-(morpholin-4-yl)-1,7-naphthyridines | Chemistry; Metallurgy | 9 | Active |
| US6127335A | Cyclic adhesion inhibitors | Human Necessities | 6 | Expired |
| US9388140B2 | Substituted benzimidazoles | Chemistry; Metallurgy | 3 | Active |
| US9993484B2 | 2-(morpholin-4-yl)-1,7-naphthyridines | Chemistry; Metallurgy | 3 | Active |
| US10772893B2 | 2-(morpholin-4-yl)-1,7-naphthyridines | Chemistry; Metallurgy | 2 | Active |
| US9284317B2 | Substituted imidazo[1,2-a]pyrazines as MPS-1 inhibitors | Chemistry; Metallurgy | 1 | Active |
| US9255100B2 | Substituted imidazopyridazines | Chemistry; Metallurgy | 1 | Active |
| US8551980B2 | Substituted triazolopyridines | Human Necessities | 1 | Active |
| US9199999B2 | Substituted imidazopyrazines | Human Necessities | 1 | Active |
| US9212184B2 | 6-thio-substituted imidazo[1,2-a]pyrazines as Mps-1 inhibitors | Human Necessities | 1 | Active |
| US9512130B2 | Substituted imidazopyridazines | Human Necessities | 0 | Active |
| US9676766B2 | Triazolopyridines | Human Necessities | 0 | Active |
| US11529356B2 | 2-(morpholin-4-yl)-1,7-naphthyridines | Chemistry; Metallurgy | 0 | Active |
| US9468642B2 | Imidazopyrazines | Chemistry; Metallurgy | 0 | Active |
| US10730856B2 | Benzimidazole derivatives as EP4 ligands | Human Necessities | 0 | Active |
| US9555022B2 | Substituted triazolopyridines | Chemistry; Metallurgy | 0 | Active |
| US10167293B2 | [8-(phenylsulfonyl)-3,8-diazabicyclo[3.2.1]oct-3-yl](1H-1,2,3-triazol-4-yl)methanones | Human Necessities | 0 | Active |
| US9512126B2 | Substituted imidazopyridazines | Human Necessities | 0 | Active |
| US10894784B2 | Heteroarylbenzimidazole compounds | Chemistry; Metallurgy | 0 | Active |
| US8729082B2 | Substituted imidazoquinoxalines | Human Necessities | 0 | Active |
| US10172814B2 | Substituted pyridyl-cycloalkyl-carboxylic acids, compositions containing them and medical uses thereof | Chemistry; Metallurgy | 0 | Active |
| US6528619B1 | Inhibitors for urokinase receptor | Chemistry; Metallurgy | 0 | Expired |
Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.