Inventor · San Diego, CA, US

Mark W. Holladay

43Patents
15h-index
91Co-inventors
84Inventor score

Filing activity: Jun 17, 1991 → Jun 28, 2017

Most-cited inventions

PatentTitleAreaCited byStatus
US5629325A 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission Chemistry; Metallurgy 60 Expired
US5346907A Amino acid analog CCK antagonists Chemistry; Metallurgy 51 Expired
US5948793A 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release Chemistry; Metallurgy 36 Expired
US8030488B2 Piperazine derivatives as stearoyl-coa desaturase inhibitors and their use as therapeutic agents Chemistry; Metallurgy 33 Active
US5914328A Heterocyclic ether compounds useful in controlling neurotransmitter release Chemistry; Metallurgy 32 Expired
US7335658B2 Pyridazine derivatives and their use as therapeutic agents Chemistry; Metallurgy 32 Expired
US5340802A Peptide analog type-B CCK receptor ligands Human Necessities 31 Expired
US5472958A 2-((nitro)phenoxymethyl) heterocyclic compounds that enhance cognitive function Human Necessities 29 Expired
US6127386A 3-Pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission Chemistry; Metallurgy 27 Expired
US6437138B1 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission Chemistry; Metallurgy 24 Expired
US8618289B2 RAF kinase modulator compounds and methods of use thereof Chemistry; Metallurgy 21 Active
US7749980B2 Non-nucleotide compositions and method for treating pain Human Necessities 19 Active
US5733912A 7A-heterocycle substituted hexahydro-1H-pyrrolizine compounds useful in controlling chemical synaptic transmission Human Necessities 18 Expired
US6265417A Potassium channel openers Chemistry; Metallurgy 16 Expired
US7456180B2 Piperazine derivatives and their use as therapeutic agents Chemistry; Metallurgy 15 Expired
US5270302A Derivatives of tetrapeptides as CCK agonists Human Necessities 14 Expired
US6593335B1 Potassium channel openers Chemistry; Metallurgy 14 Expired
US7919484B2 Combination therapy Human Necessities 9 Active
US8969587B2 RAF kinase modulator compounds and methods of use thereof Chemistry; Metallurgy 7 Active
US6133253A 3-Pyridyl enantiomers and their use as analgesics Chemistry; Metallurgy 7 Expired
US9320739B2 RAF kinase modulator compounds and methods of use thereof Chemistry; Metallurgy 6 Active
US6001849A Furopyridine, thienopyridine pyrrolopyridine useful in controlling chemical synaptic transmission Chemistry; Metallurgy 3 Expired
US9725465B2 Biaryl acetamide compounds and methods of use thereof Chemistry; Metallurgy 3 Active
US6274587A Tricyclic dihydropyrimidine potassium channel openers Chemistry; Metallurgy 3 Expired
US10829484B2 Compounds and methods for kinase modulation, and indications therefor Chemistry; Metallurgy 3 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.