Inventor · Boston, MA, US

Andreas Goutopoulos

49Patents
7h-index
65Co-inventors
72Inventor score

Filing activity: Nov 24, 1999 → Nov 4, 2020

Most-cited inventions

PatentTitleAreaCited byStatus
US8076486B2 Heteroaryl-substituted arylaminopyridine derivatives as MEK inhibitors Chemistry; Metallurgy 24 Active
US8815872B2 Macrocyclics pyrimidines as aurora kinase inhibitors Chemistry; Metallurgy 16 Active
US7956191B2 3-arylamino pyridine derivatives Chemistry; Metallurgy 15 Active
US8637532B2 Amino azaheterocyclic carboxamides Chemistry; Metallurgy 9 Active
US9624246B2 Pyridazinone macrocycles as IRAK inhibitors and uses thereof Chemistry; Metallurgy 7 Active
US9708324B2 Macrocyclic compounds as IRAK1/4 inhibitors and uses thereof Chemistry; Metallurgy 7 Active
US9073947B2 Compositions and methods for the production of pyrimidine and pyridine compounds with BTK inhibitory activity Chemistry; Metallurgy 7 Active
US8569295B2 Bicyclic urea compounds Chemistry; Metallurgy 7 Active
US8198457B2 3-arylamino pyridine derivatives Chemistry; Metallurgy 7 Active
US8524911B2 3-arylamino pyridine derivatives Chemistry; Metallurgy 6 Active
US9815836B2 Macrocyclic compounds as IRAK1/4 inhibitors and uses thereof Chemistry; Metallurgy 6 Active
US9440968B2 Substituted pyrido[3,2-d]pyrimidines for treating cancer Chemistry; Metallurgy 5 Active
US8841459B2 3-arylamino pyridine derivatives Chemistry; Metallurgy 5 Active
US8946227B2 Piperazine derivatives and methods of use Chemistry; Metallurgy 4 Active
US9181226B2 Benzamides Chemistry; Metallurgy 4 Active
US8791114B2 Dihydropyrazoles Chemistry; Metallurgy 4 Active
US9580449B2 Compositions and methods for the production of pyrimidine and pyridine compounds with BTK inhibitory activity Chemistry; Metallurgy 3 Active
US7754722B2 Piperazine derivatives and methods of use Chemistry; Metallurgy 3 Active
US9498475B2 Benzamides Chemistry; Metallurgy 3 Active
US9938262B2 Benzamides Chemistry; Metallurgy 2 Active
US9775830B2 Dihydropyrazoles Chemistry; Metallurgy 2 Active
US7161016B1 Cannabimimetic lipid amides as useful medications Chemistry; Metallurgy 2 Expired
US10016448B2 Compositions and methods for the production of pyrimidine and pyridine compounds with BTK inhibitory activity Chemistry; Metallurgy 2 Active
US8884023B2 Pyrano [3,2-D][1,3]thiazole as glycosidase inhibitors Human Necessities 2 Active
US9040560B2 Amino azaheterocyclic carboxamides Chemistry; Metallurgy 2 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.