Inventor · Caldwell, NJ, US

Stuart W. McCombie

48Patents
16h-index
62Co-inventors
84Inventor score

Filing activity: Jun 30, 1976 → Mar 26, 2008

Most-cited inventions

PatentTitleAreaCited byStatus
US5883096A Muscarinic antagonists Chemistry; Metallurgy 74 Expired
US5889006A Muscarinic antagonists Chemistry; Metallurgy 58 Expired
US6689765B2 Piperazine derivatives useful as CCR5 antagonists Chemistry; Metallurgy 49 Expired
US6066636A Muscarinic antagonists Chemistry; Metallurgy 45 Expired
US6037352A Muscarinic antagonists Chemistry; Metallurgy 44 Expired
US6391865B1 Piperazine derivatives useful as CCR5 antagonists Chemistry; Metallurgy 43 Expired
US7750158B2 Cannabinoid receptor ligands Chemistry; Metallurgy 40 Active
US6387930B1 Piperidine derivatives useful as CCR5 antagonists Chemistry; Metallurgy 34 Expired
US6294554A Muscarinic antagonists Chemistry; Metallurgy 29 Expired
US4876365A Intermediate compounds for preparing penems and carbapenems Chemistry; Metallurgy 27 Expired
US6043255A Muscarinic antagonists Chemistry; Metallurgy 23 Expired
US4078139A Process for deoxygenating secondary alcohols Chemistry; Metallurgy 20 Expired
US4582918A Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols Chemistry; Metallurgy 19 Expired
US4237051A Stereospecific production of 6- or 7-carbon-substituted-.beta.-lactams Chemistry; Metallurgy 18 Expired
US5064837A 3-substituted-1-aryl-2(H)-quinolones and their pharmaceutical compositions Chemistry; Metallurgy 17 Expired
US5318971A 3-Substituted-1-aryl-2(1H)-quinolones useful as anti-allergy and anti-inflammatory agents Chemistry; Metallurgy 17 Expired
US4973750A Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols Chemistry; Metallurgy 14 Expired
US6894063B2 Substituted urea neuropeptide Y Y5 Receptor antagonists Chemistry; Metallurgy 13 Expired
US4212859A 2'-Hydroxy-2'-desamino-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols, methods for their manufacture, method for their use as antibacterial agents, and compositions useful therefor Emerging Cross-Sectional Technologies 13 Expired
US4272439A 6-(Substituted-hydroxymethylene penams) Chemistry; Metallurgy 12 Expired
US4314942A Deprotection of allylic esters, carbonates and carbamates catalyzed by palladium compounds Chemistry; Metallurgy 11 Expired
US6288068A Muscarinic antagonists Chemistry; Metallurgy 11 Expired
US5179093A Quinoline-diones Chemistry; Metallurgy 9 Expired
US4053591A 5-Deoxy-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols, methods for their manufacture, method for their use as antibacterial agents and compositions useful therefor Emerging Cross-Sectional Technologies 8 Expired
US6946476B2 Heteroaryl urea neuropeptide Y Y5 receptor antagonists Chemistry; Metallurgy 7 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.