Inventor · Jerusalem, IL

Chaim Gilon

27Patents
9h-index
33Co-inventors
75Inventor score

Filing activity: Apr 16, 1991 → Mar 12, 2019

Most-cited inventions

PatentTitleAreaCited byStatus
US5217999A Styryl compounds which inhibit EGF receptor protein tyrosine kinase Chemistry; Metallurgy 183 Expired
US5302606A Styryl-substituted pyridyl compounds which inhibit EGF receptor tyrosine kinase Chemistry; Metallurgy 176 Expired
US5874529A Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 73 Expired
US7084244B2 Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 57 Expired
US5196446A Certain indole compounds which inhibit EGF receptor tyrosine kinase Chemistry; Metallurgy 48 Expired
US5770687A Comformationally constrained backbone cyclized somatostatin analogs Emerging Cross-Sectional Technologies 29 Expired
US5811392A Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 15 Expired
US5656655A Styryl-substituted heteroaryl compounds which inhibit EGF receptor tyrosine kinase Chemistry; Metallurgy 12 Expired
US5723575A Process for the preparation of backbone cyclic peptides Emerging Cross-Sectional Technologies 10 Expired
USRE38761E1 Styryl compounds which inhibit EGF receptor protein tyrosine kinase General 9 Expired
US5883293A Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 8 Expired
US6117974A Libraries of backbone-cyclized peptidomimetics Emerging Cross-Sectional Technologies 8 Expired
US6265375A Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 6 Expired
US5677329A Styryl-substituted monocyclic and bicyclic heteroaryl compounds which inhibit EGF receptor tyrosine kinase Chemistry; Metallurgy 4 Expired
US6407059B1 Conformationally constrained backbone cyclized peptide analogs Emerging Cross-Sectional Technologies 3 Expired
US8658603B2 Compositions and methods for inducing an immune response Human Necessities 2 Active
US5990277A Semipeptoid farnesyl protein transferase inhibitors and analogs thereof Human Necessities 1 Expired
US10155790B2 Antagonists of neurokinin B in fish reproduction Emerging Cross-Sectional Technologies 1 Active
US10793614B2 Antagonists of fish reproduction Human Necessities 0 Active
US11261215B2 Somatostatin prodrugs Human Necessities 0 Active
US10662225B2 Backbone cyclized inhibitory peptides of myeloid differentiation factor 88 (MyD88) Human Necessities 0 Active
US6664368B1 Inhibition of nuclear import by backbone cyclic peptide analogs Chemistry; Metallurgy 0 Expired
US11267846B2 High shear solid phase synthesis Performing Operations; Transporting 0 Active
US8198218B2 Heterocyclic compounds, combinatorial libraries thereof and methods of selecting drug leads Chemistry; Metallurgy 0 Active
US11965041B2 N-methylated cyclic peptides and their prodrugs Human Necessities 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.