Inventor · Wuppertal, DE

Johannes-Peter Stasch

153Patents
26h-index
153Co-inventors
93Inventor score

Filing activity: Mar 6, 1987 → Aug 18, 2022

Most-cited inventions

PatentTitleAreaCited byStatus
US7173037B2 Carbamate-substituted pyrazolopyridines Human Necessities 122 Expired
US6743798B1 Substituted pyrazole derivatives condensed with six-membered heterocyclic rings Human Necessities 116 Expired
US6833364B1 Substituted pyrazole derivatives Chemistry; Metallurgy 103 Expired
US6693102B2 Pyridine-substituted pyrazolopyridine derivatives Human Necessities 90 Expired
US6180656A Use of condensated (hetaryl-substituted) 1-benzal-3-pyrazol derivates for treating special diseases of the cardiovascular and the central nervous systems Human Necessities 79 Expired
US6864287B1 Derivatives of dicarboxylic acid having pharmaceutical properties Chemistry; Metallurgy 57 Expired
US5407948A Substituted mono- and bipyridylmethylpyridones Human Necessities 56 Expired
US6451805B1 Substituted pyrazole derivatives for the treatment of cardiocirculatory diseases Chemistry; Metallurgy 55 Expired
US7674825B2 Dicarboxylic acid derivatives with pharmaceutical properties Chemistry; Metallurgy 49 Active
US8420656B2 Substituted 5-fluoro-1H-pyrazolopyridines and their use Chemistry; Metallurgy 48 Active
US6166027A Heterocyclylmethyl-substituted pyrazole derivatives and their use for treating cardiovascular diseases Chemistry; Metallurgy 48 Expired
US5356911A Substituted biphenylpyridones Human Necessities 46 Expired
US6903089B1 Lactam-substituted pyrazolopyridine derivatives Human Necessities 44 Expired
US5254543A Sulphonylbenzyl-substituted pyridones which are angiotension II receptor antagonists Chemistry; Metallurgy 42 Expired
US7705043B2 Substituted aminodicarboxylic acid derivatives having pharmaceutical properties Chemistry; Metallurgy 36 Active
US8309551B2 Pyrazolopyridine, indazole, imidazopyridine, imidazopyrimidine, pyrazolopyrazine and pyrazolopyridine derivatives as stimulators of guanylate cyclase for cardiovascular disorders Chemistry; Metallurgy 36 Active
US5395840A Heterocyclically substituted phenyl-cyclohexane-carboxylic acid derivatives Human Necessities 36 Expired
US7078417B2 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use as cardiovascular preparations Chemistry; Metallurgy 35 Expired
US7087644B1 Derivatives of dicarboxylic acid having pharmaceutical properties Chemistry; Metallurgy 35 Expired
US7129255B2 Substituted 2-carba-3,5-dicyano-4-aryl-6-aminopyridines and the use of the same as selective ligands of the adenosine receptor Chemistry; Metallurgy 33 Expired
US7045631B2 Substituted 2-thio-3, 5-dicyano-4-phenyl-6-aminopyridines and their use as adenosine receptor-selective ligands Chemistry; Metallurgy 33 Expired
US7109218B2 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same Chemistry; Metallurgy 33 Expired
US9216978B2 Ring-fused pyrimidines and triazines and use thereof for the treatment and/or prophylaxis of cardiovascular diseases Chemistry; Metallurgy 31 Active
US7410973B2 4-amino-substituted pyrimidine derivatives Human Necessities 29 Expired
US6919345B2 Sulfonate substituted pyrazol pyridine derivatives Human Necessities 28 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.