Inventor · Del Mar, CA, US

Mark D. Erion

61Patents
20h-index
50Co-inventors
91Inventor score

Filing activity: Oct 31, 1989 → May 6, 2022

Most-cited inventions

PatentTitleAreaCited byStatus
US6312662A Prodrugs phosphorus-containing compounds Emerging Cross-Sectional Technologies 195 Expired
US5294632A Phosphono/biaryl substituted dipetide derivatives Human Necessities 150 Expired
US5155100A Phosphono/biaryl substituted dipeptide derivatives Human Necessities 136 Expired
US6489476B1 Heteroaromatic compounds containing a phosphonate group that are inhibitors of fructose-1,6-bisphosphatase Chemistry; Metallurgy 115 Expired
US5506347A Lyxofuranosyl analogues of adenosine Chemistry; Metallurgy 115 Expired
US5646128A Methods for treating adenosine kinase related conditions Chemistry; Metallurgy 114 Expired
US5763596A C-4' modified adenosine kinase inhibitors Chemistry; Metallurgy 101 Expired
US5674998A C-4' modified adenosine kinase inhibitors Chemistry; Metallurgy 100 Expired
US5763597A Orally active adenosine kinase inhibitors Chemistry; Metallurgy 99 Expired
US5795977A Water soluble adenosine kinase inhibitors Chemistry; Metallurgy 90 Expired
US6752981B1 Prodrugs for liver specific drug delivery Emerging Cross-Sectional Technologies 51 Expired
US6054587A Indole and azaindole inhibitors of fructose-1,6-bisphosphatase Chemistry; Metallurgy 50 Expired
US6399782B1 Benzimidazole inhibitors of fructose 1,6-bisphosphatase Chemistry; Metallurgy 39 Expired
US6110903A Benzimidazole inhibitors of fructose 1,6-bisphosphatase Chemistry; Metallurgy 39 Expired
US6284748A Purine inhibitors of fructose 1,6-bisphosphatase Chemistry; Metallurgy 38 Expired
US6946115B2 Prodrugs for phosphorus-containing compounds Emerging Cross-Sectional Technologies 36 Expired
US6294672A Indole and azaindole inhibitors of Fructose-1,6-biphosphatase Chemistry; Metallurgy 30 Expired
US5726302A Water soluble adenosine kinase inhibitors Chemistry; Metallurgy 22 Expired
US5008270A 2-amino-7-(heterocyclomethyl)-3H,5H-pyrrolo[3,2-d]pyrimidin-4-ones and pharmaceutical uses and compositions containing the same Chemistry; Metallurgy 21 Expired
US6756360B1 Combination of FBPase inhibitors and insulin sensitizers for the treatment of diabetes Human Necessities 20 Expired
US4985434A 7-substituted derivatives of 2-amino-3H,5H-pyrrolo(3,2-d)pyrimidin-4-ones and pharamceutical uses and compositions containing the same Chemistry; Metallurgy 20 Expired
US5008265A 2-amino-7-(alicyclomethyl)-3H,5H,-pyrrolo[3,2-d]pyrimidin-4-ones and pharmaceutical uses and compositions containing the same Chemistry; Metallurgy 20 Expired
US4985433A 2-amino-7-(pyridinylmethyl)-3H,5H-pyrrolo[3,2-d]pyrimidin-4-ones and pharmaceutical uses and compositions containing the same Chemistry; Metallurgy 19 Expired
US5189039A 7-disubstituted-methyl-4-oxo-3H,5H-pyrrolo[3,2d]pyrimidine and pharmaceutical uses and compositions containing the same Chemistry; Metallurgy 16 Expired
US7514419B2 Phosphorus-containing thyromimetics Chemistry; Metallurgy 15 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.