Inventor · Westfield, NJ, US

William W. Leong

36Patents
7h-index
83Co-inventors
72Inventor score

Filing activity: Jul 8, 1994 → Sep 14, 2023

Most-cited inventions

PatentTitleAreaCited byStatus
US8569494B2 Methods of synthesis and purification of heteroaryl compounds Chemistry; Metallurgy 19 Active
US5486625A Process for the preparation of chiral intermediates useful for the synthesis of antifungal agents Chemistry; Metallurgy 18 Expired
US9309220B2 Processes for the preparation of (S)-3-(4- (4-(morpholinomethyl)benzyl)oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione and pharmaceutically acceptable forms thereof Chemistry; Metallurgy 11 Active
US9359364B2 Pharmaceutical formulations, processes, solid forms and methods of use relating to 1-ethyl-7-(2-methyl-6-(1H-1,2,4-triazol-3-yl)pyridin-3-yl)-3,4-dihydropyrazino[2,3-b] pyrazin-2(1H)-one Chemistry; Metallurgy 11 Active
US9403829B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use Human Necessities 10 Active
US5625064A Process for the preparation of triazolones Chemistry; Metallurgy 8 Expired
US6958337B2 Crystalline antifungal polymorph Chemistry; Metallurgy 8 Expired
US8802685B2 Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses Human Necessities 7 Active
US8686135B2 Methods of synthesis and purification of heteroaryl compounds Chemistry; Metallurgy 7 Active
US9067912B2 Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidine-2,8-dione Chemistry; Metallurgy 5 Active
US6713481B1 Crystalline antifungal polymorph Chemistry; Metallurgy 4 Expired
US9079900B2 Methods of synthesis and purification of heteroaryl compounds Chemistry; Metallurgy 4 Active
US10220050B2 Isotopologues of 5-azacytidine Human Necessities 3 Active
US9126906B2 Asymmetric synthetic processes for the preparation of aminosulfone compounds Chemistry; Metallurgy 3 Active
US9751853B2 Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses Human Necessities 3 Active
US10463683B2 Isotopologues of 5-azacytidine Human Necessities 3 Active
US9249121B2 Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses Human Necessities 2 Active
US10646503B2 Isotopologues of 5-azacytidine Human Necessities 2 Active
US9682952B2 Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl) piperidine-2-6-dione and methods of preparation thereof Human Necessities 2 Active
US6936718B2 Preparation of rotamer mixtures of pharmaceutical salts Human Necessities 2 Expired
US6992189B2 Synthesis of piperidine and piperazine compounds as CCR5 antagonists Chemistry; Metallurgy 1 Expired
US9975872B2 Processes for the preparation of (s)-3-(4-((4-(morpholinomethyl)benzyl)oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione and pharmaceutically acceptable forms thereof Chemistry; Metallurgy 1 Active
US9303014B2 Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidine-2,6-dione Chemistry; Metallurgy 1 Active
US9969713B2 Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses Human Necessities 1 Active
US9266858B2 Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidine-2,6-dione Chemistry; Metallurgy 1 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.