Inventor · San Diego, CA, US

Alexander Chucholowski

35Patents
11h-index
74Co-inventors
78Inventor score

Filing activity: Dec 10, 1987 → Mar 1, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US6242644A N-(4-carbamimidoyl-phenyl)-glycine derivatives Chemistry; Metallurgy 45 Expired
US5830920A Sulfuric acid esters of sugar alcohols Chemistry; Metallurgy 30 Expired
US8815906B2 Tyrosine kinase inhibitors Human Necessities 29 Active
US6506744B1 Benzazepinone-derivatives Chemistry; Metallurgy 27 Expired
US4906624A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis Chemistry; Metallurgy 27 Expired
US4950675A Pyridine di-mevalono-lactones as inhibitors of cholesterol biosynthesis Chemistry; Metallurgy 20 Expired
US9562019B2 Substituted pyridazines as EGFR and/or KRAS inhibitors Chemistry; Metallurgy 19 Active
US5153226A Acat inhibitors for treating hypocholesterolemia Chemistry; Metallurgy 19 Expired
US4997837A 6-(((substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis Chemistry; Metallurgy 18 Expired
US5521160A Sulfuric acid esters of sugar alcohols Chemistry; Metallurgy 17 Expired
US4929620A 5-pyrimidinyl-3,5-dihydroxy-6-heptenoic acid compounds useful as inhibitors of cholesterol biosynthesis Chemistry; Metallurgy 14 Expired
US5767268A Sulfuric acid esters of amino sugars Chemistry; Metallurgy 10 Expired
US8063225B2 Tricyclic compound derivatives useful in the treatment of neoplastic diseases, inflammatory disorders and immunomodulatory disorders Human Necessities 10 Active
US8629147B2 Heterocyclic compounds useful in the treatment of neoplastic diseases, inflammatory disorders and immunomodulatory disorders Chemistry; Metallurgy 9 Active
US4868185A 6-[[Substituted)pyrimidinyl)ethyl]- and ethenyl]tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis Chemistry; Metallurgy 9 Expired
US7102007B2 Dihydroindole and tetrahydroquinoline derivatives Chemistry; Metallurgy 5 Expired
US6790860B2 Pyrrolidine derivatives Emerging Cross-Sectional Technologies 5 Expired
US9884127B2 Drug-conjugates, conjugation methods, and uses thereof Chemistry; Metallurgy 3 Active
US6706751B2 Dihydroindole and tetrahydroquinoline derivatives Chemistry; Metallurgy 3 Expired
US6683215B2 N-(4-carbamimidoyl-phenyl)-glycine derivatives Chemistry; Metallurgy 2 Expired
US7189756B2 Pyrrolidine derivatives Emerging Cross-Sectional Technologies 2 Expired
US5073565A Tetrazole ureas and thioureas and their use as ACAT inhibitors Chemistry; Metallurgy 2 Expired
US6858651B2 2,3-oxidosqualene-lanosterol cyclase inhibitors Chemistry; Metallurgy 2 Expired
US6541638B2 Pyrrolidine derivatives Chemistry; Metallurgy 2 Expired
US6476264B2 N-(4-carbamimidoyl-phenyl)-glycine derivatives Chemistry; Metallurgy 2 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.