Inventor · Ulm, DE

Alexander Pautsch

29Patents
13h-index
62Co-inventors
84Inventor score

Filing activity: Oct 16, 2002 → Nov 4, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US7173028B2 Pyrimidine derivatives Chemistry; Metallurgy 78 Expired
US8211923B2 Substituted arylsulfonylaminomethylphosphonic acid derivatives, their preparation and their use in the treatment of type I and II diabetes mellitus Chemistry; Metallurgy 50 Active
US8987249B2 Substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C Emerging Cross-Sectional Technologies 42 Active
US9073869B2 Method of using substituted 2-Aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Chemistry; Metallurgy 18 Active
US8999975B2 Substituted N- [1-cyano-2- (phenyl) ethyl] -2-azabicyclo [2.2.1] heptane-3-carboxamide inhibitors of cathepsin C Emerging Cross-Sectional Technologies 18 Active
US8889708B2 Substituted bicyclic 1-carboxylic-acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Emerging Cross-Sectional Technologies 17 Active
US8877775B2 Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Chemistry; Metallurgy 17 Active
USRE47636E1 Substituted spirocycles General 16 Active
US10238633B2 Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C Emerging Cross-Sectional Technologies 16 Active
US9713606B2 Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C Emerging Cross-Sectional Technologies 16 Active
US8871783B2 Substituted 2-aza-bicyclo[2.2.1]heptane-3-carboxylic acid (cyano-methyl)-amides inhibitors of cathepsin C Chemistry; Metallurgy 15 Active
US9879026B2 Substituted spirocycles Chemistry; Metallurgy 15 Active
US9440960B2 Substituted oxetanes and their use as inhibitors of cathepsin C Chemistry; Metallurgy 15 Active
US7709480B2 Pyrimidine derivatives Chemistry; Metallurgy 9 Active
US8420630B2 Pyrimidine derivatives Chemistry; Metallurgy 6 Active
US7517995B2 Thiazolyl-dihydro-cyclopentapyrazole Human Necessities 4 Active
US10640486B2 Heteroarylcarboxamide derivatives as plasma kallikrein inhibitors Human Necessities 3 Active
US10399961B2 Heteroarylcarboxamide derivatives as plasma kallikrein inhibitors Chemistry; Metallurgy 3 Active
US9540373B2 Substituted spirocycles Chemistry; Metallurgy 2 Active
US7691868B2 Thiazolyl-dihydro-quinazoline Human Necessities 1 Active
US8232286B2 Inhibitors of PI3-kinases Chemistry; Metallurgy 1 Active
US8410100B2 Pteridinone derivatives as PI3-kinases inhibitors Human Necessities 0 Active
US8334378B2 Thiazolyl-dihydro-quinazoline compounds and processes for preparing same Human Necessities 0 Active
US8357689B2 Substituted arylsulfonylaminomethylphosphonic acid derivatives, their preparation and their use in the treatment of type I and II diabetes mellitus Chemistry; Metallurgy 0 Active
US11691960B2 2-[thiophen-2-yl)formamido]-N-(phenyl)-2-methylpropanamide derivatives and the use thereof as medicament Human Necessities 0 Active

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.