Inventor · Hofheim, DE

Holger Heitsch

34Patents
9h-index
53Co-inventors
78Inventor score

Filing activity: Sep 10, 1990 → Apr 4, 2011

Most-cited inventions

PatentTitleAreaCited byStatus
US5236943A Method for the treatment of cardiac and of vascular hypertrophy and hyperplasia Human Necessities 22 Expired
US5604251A Imidazole derivatives with a biphenylsulfonylurea or biphenylsulfonylurethane side chain and their use as angitensin II receptors Chemistry; Metallurgy 16 Expired
US6235766A 1-(p-thienylbenzyl)imidazoles as agonists of angiotensin (1-7) receptors, processes for their preparation, their use, and pharmaceutical preparations comprising them Human Necessities 15 Expired
US6511989B2 Acylaminoalkyl-substituted benzenesulfonamide derivatives, their preparation, their use and pharmaceutical preparations comprising them Chemistry; Metallurgy 14 Expired
US5635525A Benzimidazole derivatives as angiotensin II receptor antagonists, pharmacticals, and treatment of hypertension therewith Chemistry; Metallurgy 13 Expired
US7919628B2 CXCR2 inhibitors Chemistry; Metallurgy 12 Active
US5786365A Use of nonpeptide bradykinin antagonists for the treatment and prevention of chronic fibrogenetic liver disorders, acute liver disorders and the complications associated therewith Human Necessities 12 Expired
US5444068A Imidazopyridine derivatives as angiotensin II receptor antagonists, pharmaceuticals, and treatment of hypertension therewith Chemistry; Metallurgy 12 Expired
US5952346A Use of non-peptide bradykinin antagonists for the treatment or prevention of Alzheimer's disease Human Necessities 10 Expired
US5475004A Angiotensin II receptor antagonists for the treatment and prophylaxis of coronary heart disease Human Necessities 9 Expired
US5612365A Angiotensin II receptor antagonists for the treatment and prophylaxis of coronary heart disease Human Necessities 8 Expired
US6211196A Benzyloxy-substituted, fused N-heterocycles, processes for their preparation, and their use as bradykinin receptor antagonists Chemistry; Metallurgy 8 Expired
US6429222B2 1-(p-thienylbenzyl)imidazoles as agonists of angiotensin (1-7) receptors, processes for their preparation, their use, and pharmaceutical preparations comprising them Human Necessities 8 Expired
US5468764A Angiotensin II receptor antagonists for the treatment of disturbances in cardiac rhythm Human Necessities 7 Expired
US6984660B2 P-thienylbenzylamides as agonists of angiotensin-(1-7) receptors, and methods of their preparation and use Chemistry; Metallurgy 7 Expired
US5527919A Process for the preparation of 1-[(1,1'-biphenyl]-4-YL]-methyl-1H-imidazole-5-carboxylic acids Chemistry; Metallurgy 7 Expired
US5859025A Fluoroalkyl- and fluoroalkoxy-substituted heterocyclic bradykinin antagonists, process for their preparation, and their use Human Necessities 6 Expired
US6462024B1 Use of inhibitors of the sodium-hydrogen exchanger for the production of a medicament for decreasing undesired effects of substrates of the heart Human Necessities 6 Expired
US6538144B2 P-thienylbenzylamides as agonists of angiotensin-(1-7) receptors, and methods of their preparation and use Chemistry; Metallurgy 5 Expired
US5834500A Sulfur-containing heterocyclic bradykinin antagonists, process for their preparation, and their use Chemistry; Metallurgy 4 Expired
US6414030B1 Use of benzenesulfonyl(thio)ureas for the treatment and prophylaxis of dysfunctions of the autonomous nervous system and use of benzenesulfonyl(thio)ureas in combination with beta-receptors blockers Chemistry; Metallurgy 3 Expired
US8283479B2 CXCR2 inhibitors Chemistry; Metallurgy 2 Active
US8044208B2 Imidazole derivatives as inhibitors of TAFIa Chemistry; Metallurgy 2 Active
US8710232B2 Imidazole derivatives used as TAFIa inhibitors Chemistry; Metallurgy 2 Active
US6979532B2 Process for identifying substances which modulate the activity of hyperpolarization-activated cation channels Physics 2 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.