Inventor · Warthausen, DE

Michael Entzeroth

24Patents
13h-index
36Co-inventors
81Inventor score

Filing activity: Jun 20, 1989 → Nov 19, 2015

Most-cited inventions

PatentTitleAreaCited byStatus
US5591762A Benzimidazoles useful as angiotensin-11 antagonists Chemistry; Metallurgy 139 Expired
US6344449B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production Emerging Cross-Sectional Technologies 73 Expired
US5602127A (Alkanesultam-1-yl)-benzimidazol-1-yl)-1yl)-methyl-biphenyls useful as angiotensin-II antagonists Chemistry; Metallurgy 70 Expired
US5594003A Tetrahydroimidazo[1,2-a]pyridin-2-yl-(benzimidazol-1-yl)-methyl-biph enyls useful as angiotensin-II antagonists Chemistry; Metallurgy 69 Expired
US5614519A (1-(2,3 or 4-N-morpholinoalkyl)-imidazol-4-yl)-benizimidazol-1-yl-methyl]-biphenyls useful as angiotensin-II antagonists Chemistry; Metallurgy 67 Expired
US5864043A Benzimidazoles, medicaments containing these compounds and processes for their preparation Chemistry; Metallurgy 55 Expired
US5385925A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 31 Expired
US5565469A Benzimidazoles and pharmaceutical compositions containing them Chemistry; Metallurgy 24 Expired
US7498325B2 Modified amino acids, pharmaceuticals containing these compounds and method for their production Physics 19 Expired
US5684029A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 18 Expired
US5587393A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 17 Expired
US5519138A Phenylalkyl derivatives, with pharmaceutical activity Chemistry; Metallurgy 13 Expired
US6114390A Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them Human Necessities 13 Expired
US5135932A 2-hydroxypropylamino-alkyl-benzimidazoly-5-yl derivatives and their use in the treatment of heart disease Chemistry; Metallurgy 13 Expired
US5459147A Substituted benzimidazolyl derivatives and pharmaceutical compositions containing these compounds Chemistry; Metallurgy 9 Expired
US5616620A Amino acid derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of obesity Chemistry; Metallurgy 9 Expired
US5541229A Benzimidazoles and medicaments containing these compounds Chemistry; Metallurgy 9 Expired
US5807875A Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 6 Expired
US5068325A 4,5,7,8-tetrahydro-6H-thiazolo[5,4-d]azepines, their preparation and their use as pharmaceutical compositions Human Necessities 4 Expired
US5270322A Imidazo[1,2-a]pyridines, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 3 Expired
US5521177A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them Chemistry; Metallurgy 1 Expired
US5641772A Condensed diazepinones, processes for preparing them and agents containing these compounds for treating diseases of the central nervous system and for promoting cerebral blood circulation Chemistry; Metallurgy 0 Expired
US10414728B2 Use of tetrahydropyridines in the treatment of sodium channel related disease and disorders Emerging Cross-Sectional Technologies 0 Active
US5610155A Condensed diazepinones, processes for preparing them and agents containing these compounds for treating diseases of the central nervous system and for promoting cerebral blood circulation Chemistry; Metallurgy 0 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.