Inventor · Pleasant Prairie, WI, US

Daryl Sauer

22Patents
6h-index
53Co-inventors
72Inventor score

Filing activity: Mar 9, 1994 → Nov 12, 2021

Most-cited inventions

PatentTitleAreaCited byStatus
US6020521A Macrolide LHRH antagonists Chemistry; Metallurgy 25 Expired
US7902379B2 Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them Chemistry; Metallurgy 18 Expired
US8350055B2 Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them Chemistry; Metallurgy 15 Active
US8183250B2 Potent PARP inhibitors Human Necessities 12 Active
US7910742B2 Survivin inhibitors Chemistry; Metallurgy 7 Active
US5955440A Macrolide LHRH antagonists Human Necessities 6 Expired
US5508383A Cyclic peptide LHRH antagonists Human Necessities 5 Expired
US5491217A LHRH antagonists having modified aminoacyl residues at positions 5 and 6 Human Necessities 4 Expired
US7320979B2 N-[(piperazinyl)hetaryl]arylsulfonamide compounds Chemistry; Metallurgy 3 Expired
US8445686B2 4-(4-pyridinyl)-benzamides and their use as rock activity modulators Chemistry; Metallurgy 3 Active
US6495562B1 Naphthamidine urokinase inhibitors Chemistry; Metallurgy 2 Expired
US9242933B2 Heterocyclic compounds as positive modulators of metabotropic glutamate receptor 2 (mGlu2 receptor) Chemistry; Metallurgy 2 Active
US8580842B2 Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them Chemistry; Metallurgy 2 Active
US9487505B2 Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them Chemistry; Metallurgy 1 Active
US6387885B1 3′,3′-N-bis-desmethyl-3′-N-cycloalkyl erythromycin derivatives as LHRH antagonists Chemistry; Metallurgy 1 Expired
US8895749B2 4-(4-pyridinyl)-benzamides and their use as rock activity modulators Chemistry; Metallurgy 1 Active
US8476275B2 N-[piperazinyl hetaryl]arylsufonamide compounds with affinity for the dopamine D3 receptor Chemistry; Metallurgy 0 Active
US8114875B2 Substituted N-heterocyclic compounds and their use as dopamine D3 receptor ligands Chemistry; Metallurgy 0 Active
US11807600B2 Synthesis of novel ketone body analogs for use as a nutritional supplement Chemistry; Metallurgy 0 Active
US7592466B2 Ureas having antiangiogenic activity Chemistry; Metallurgy 0 Active
US8207160B2 Tetrahydrobenzazepines and their use in he modulation of the dopamine D3 receptor Chemistry; Metallurgy 0 Active
US5972898A 3',3-N-bis-substituted macrolide LHRH antagonists Human Necessities 0 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.