Inventor · Bremen, DE

Hans Briem

55Patents
11h-index
139Co-inventors
81Inventor score

Filing activity: Jun 7, 1995 → Aug 21, 2020

Most-cited inventions

PatentTitleAreaCited byStatus
US7312225B2 Macrocyclic pyrimidines, their production and use as pharmaceutical agents Chemistry; Metallurgy 57 Expired
US7166599B2 Trisubstituted pyrimidines Chemistry; Metallurgy 30 Expired
US5710155A Arylglycinamide derivatives, processes for the manufacture thereof and pharmaceutical compositions containing these compounds Chemistry; Metallurgy 19 Expired
US5696123A Neurokinin antagonists Chemistry; Metallurgy 18 Expired
US9549932B2 2-(morpholin-4-yl)-1,7-naphthyridines Chemistry; Metallurgy 16 Active
US5861509A Arylglycinamide derivatives and pharmaceutical compositions containing these compounds Chemistry; Metallurgy 16 Expired
US5985881A Neurokinin antagonists Chemistry; Metallurgy 15 Expired
US5708006A Neurokinin antagonists Chemistry; Metallurgy 15 Expired
US6235732A Neurokinin antagonists Chemistry; Metallurgy 13 Expired
US7504410B2 Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents Chemistry; Metallurgy 13 Expired
US6191135A Neurokinin antagonists Chemistry; Metallurgy 13 Expired
US6512000B1 Aminocarbonyl-substituted benzimidazoles having tryptase-inhibitory activity Chemistry; Metallurgy 5 Expired
US7825128B2 Sulfoximine-substituted pyrimidines, processes for production thereof and use thereof as drugs Chemistry; Metallurgy 5 Active
US9643953B2 Substituted benzylpyrazoles Chemistry; Metallurgy 4 Active
US9682974B2 Heteroaryl substituted pyrazoles Chemistry; Metallurgy 4 Active
US6124296A Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds Chemistry; Metallurgy 3 Expired
US9765058B2 Substituted benzylpyrazoles Human Necessities 3 Active
US9745285B2 Heteroaryl substituted pyrazoles Chemistry; Metallurgy 3 Active
US6294556A Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds Chemistry; Metallurgy 3 Expired
US6365584B1 Arylysulphonamide-substituted benzimidazoles having tryptase-inhibiting activity Chemistry; Metallurgy 3 Expired
US9993484B2 2-(morpholin-4-yl)-1,7-naphthyridines Chemistry; Metallurgy 3 Active
US10772893B2 2-(morpholin-4-yl)-1,7-naphthyridines Chemistry; Metallurgy 2 Active
US6514969B2 &bgr;-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions Human Necessities 2 Expired
US6251909A Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds Chemistry; Metallurgy 2 Expired
US6121262A Arylglycinamide derivatives, processes for the manufacture thereof and pharmaceutical compositions containing these compounds Chemistry; Metallurgy 2 Expired

Source: USPTO / EPO open patent data. Inventor disambiguation is heuristic; counts are objective bibliographic measures.